| Compound ID | Pharmacological profile | Compound name | Binding data | Activity data | Bibliographic ref | Cross-reactivity | |
| CID123976 | agonist | 27-hydroxycholesterol | PMID: 20203100 | ||||
| CID167685 | agonist | 22(R)-hydroxycholesterol | EC50 = 20-40 nM | PMID: 20203100 | |||
| CID168038 | agonist | 22(S)-hydroxycholesterol | PMID: 20203100 | ||||
| CID17980288 | agonist | SR1078 | PMID: 20735016 | ROR_alpha | |||
| CID65094 | agonist | 25-hydroxycholesterol | EC50 = 20-40 nM | PMID: 20203100 | |||
| ZINC02386791 | antagonist | cerebrosterol | Ki = 25 nM | IC50 = 1300 nM | PMID: 20211758 | 
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| ZINC02557432 | agonist | cholesterol | EC50 = 200 nM | PMID: 20203100 | ROR_alpha | ||
| ZINC04096158 | antagonist | 7-alpha-hydroxycholesterol | IC50 = 1.6 µM | PMID: 19965867 | ROR_alpha | ||
| ZINC04096811 | agonist | 20-alpha-hydroxycholesterol | EC50 = 20-40 nM | PMID: 20203100 | |||
| ZINC05758789 | antagonist | 7-keto-cholesterol | IC50 = 0.6 µM | PMID: 19965867 | ROR_alpha | ||
| ZINC05758832 | antagonist | 7-beta-hydroxycholesterol | IC50 = 2.2 µM | PMID: 19965867 | ROR_alpha |