| Compound ID | Pharmacological profile | Compound name | Binding data | Activity data | Bibliographic ref | Cross-reactiviy | |
| CHEMBL260419 | antagonist | Compound 14 | IC50 = 21.5 +/- 3.5 µM | PMID: 18374567 | |||
| CHEMBL261114 | antagonist | Compound 25 | IC50 = 3.22 +/- 0.34 µM | PMID: 18374567 | SF1 | ||
| CHEMBL261115 | antagonist | Compound 26 | IC50 = 1.68 +/- 0.43 µM | PMID: 18374567 | SF1 | ||
| CHEMBL265938 | antagonist | Compound 33 | IC50 = 22.6 +/- 2.0 µM | PMID: 18374567 | SF1 | ||
| CHEMBL408947 | antagonist | Compound 34 | IC50 = 25.0 +/- 3.9 µM | PMID: 18374567 | SF1 | ||
| CHEMBL411889 | antagonist | Compound 35 | IC50 = 30.7 +/- 10.7 µM | PMID: 18374567 | SF1 | ||
| CHEMBL412079 | antagonist | Compound 30 | IC50 = 36.5 +/- 6.0 µM | PMID: 18374567 | SF1 | ||
| CID17980288 | agonist | SR1078 | PMID: 20735016 | ROR_gamma | |||
| CID23640022 | antagonist | Compound 36 | IC50 = 16.5 +/- 2.2 µM | PMID: 18374567 | |||
| CID23640023 | antagonist | Compound 37 | IC50 = 23.1 +/- 6.1 µM | PMID: 18374567 | |||
| ZINC02386791 | antagonist | cerebrosterol | Ki = 27 nM | IC50 = 620 nM | PMID: 20211758 | 
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| ZINC02557432 | agonist | cholesterol | PMID: 12467577 | ROR_gamma | |||
| ZINC04096158 | antagonist | 7-alpha-hydroxycholesterol | IC50 = 1.3 µM | PMID: 19965867 | ROR_gamma | ||
| ZINC05758789 | antagonist | 7-keto-cholesterol | IC50 = 1.4 µM | PMID: 19965867 | ROR_gamma | ||
| ZINC05758832 | antagonist | 7-beta-hydroxycholesterol | IC50 = 0.7 µM | PMID: 19965867 | ROR_gamma | ||
| ZINC12494196 | agonist | cholesterol sulfate | PMID: 12467577 |