Compound ID Pharmacological profile Compound name Binding data Activity data Bibliographic ref Cross-reactivity
CHEMBL468623 agonist Compound 10 EC50 = 520 nM PMID: 19058965
ZINC00006827 agonist Compound 11b Relative IC50 = 13 Relative EC30 =0.19 PMID: 10762038 RAR_beta
ZINC00007543 agonist Compound 1b Relative IC50 = 1.4 +/- 0.3 Relative EC30 = 0.37 +/- 0.02 PMID: 10956201 RAR_beta
ZINC00017723 agonist Compound 11a IC50 = 24 Relative EC30 = 2.8 PMID: 10762039
ZINC00538415 agonist AM80 IC50 = 124 nnM EC50 = 45 +/- 28 nM PMID: 7791761
ZINC00583260 agonist Compound 1f Relative IC50 = 1.9 +/- 0.4 Relative EC30 = 0.29 +/- 0.04 PMID: 10956201 RAR_beta
ZINC00840991 agonist Compound 20b Relative IC50 = 19 +/- 5 ED30 = 0.21 +/- 0.02 nM PMID: 10669568 RAR_gamma
ZINC01397300 agonist Compound 1 EC50 = 4µM PMID: 11405897
ZINC01483343 agonist Compound 16 EC50 = 225 nM PMID: 10543887 RAR_gamma
ZINC01532939 agonist SR11004 EC50 = 4500 nM PMID: 7650690 
RAR_beta
ZINC01533168 agonist Compound 190121 Kd = 135 nM EC50 = 435 nM PMID: 11277515
RAR_beta
ZINC01538323 antagonist Ro-41-5253 IC50 = 60 nM PMID: 8264595
ZINC01538326 antagonist Ro 46-5471 IC50 = 27 nM PMID: 8264595
ZINC01539148 antagonist ER27191 IC50 = 0.34 nM IC50 = 4.9 nM PMID: 7636879 RAR_gamma
ZINC01539149 antagonist Compound 55 IC50 = 0.91 nM IC50 = 1.3 nM PMID: 7636879 RAR_gamma
ZINC01539150 antagonist Compound 40 IC50 = 0.16 nM IC50 = 5.6 nM PMID: 7636879 RAR_gamma
ZINC01539151 antagonist Compound 4 IC50 = 16 nM IC50 = 0.12 µM PMID: 7636879 RAR_gamma
ZINC01542199 agonist Tazarotene EC50 = 63 nM PMID: 19058965
RAR_beta
ZINC01543482 antagonist AGN193109 Kd = 16 +/- 5 IC50 = 9 +/- 1 PMID: 8798442 RAR_gamma
ZINC01550227 antagonist Compound 1 Kd = 148 nM IC50 = 210 nM PMID: 11277517
ZINC01550228 antagonist Compound 2 Kd = 136 nM Ic50 = 220 nM PMID: 11277517
ZINC01550229 antagonist Compound 3 Kd = 875 nM IC50 = 350 nM PMID: 11277517
ZINC01550230 antagonist Compound 4 Kd = 252 nM IC50 = 129 nM PMID: 11277517
ZINC01550918 agonist Compound 14 EC50 = 1400 nM PMID: 9733501
RAR_gamma
ZINC01891052 agonist LG100567 Ki = 63.5 +/- 8.5 nM EC50 = 65 +/- 12 nM PMID: 8709094
RAR_beta
ZINC01891456 agonist Compound 37 EC50= 63 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC01891459 agonist Compound 33 EC50= 25 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC01891905 agonist AGN193835 Kd = 4.4 +/- 2.3 nM PMID: 8759622 RAR_beta
ZINC01893319 antagonist BMS614 Ki = 2.5 nM PMID: 10421757
ZINC01895357 antagonist Compound 5 Kd = 1.5 +/- 0.8 nM PMID: 9258350
RAR_beta
ZINC01895361 antagonist Compound 1 Kd = 27 +/- 15 nM PMID: 9258350
RAR_beta
ZINC01895365 antagonist Compound 2 Kd = 5.7 +/- 0.9 nM PMID: 9258350
RAR_beta
ZINC01895368 antagonist Compound 3 Kd = 32 +/- 15 nM PMID: 9258350 RAR_beta
ZINC01895370 antagonist Compound 4 Kd = 2.8 +/- 1.1 nM PMID: 9258350
RAR_beta
ZINC01896358 antagonist Compound 2b Kd = 17 nM IC50 = 6.5 nM PMID: 10201840
RAR_beta
ZINC01909562 agonist AGN195183 Kd = 3 nM EC50 = 200 nM PMID: 12372520
ZINC01996688 antagonist Compound 3a Kd = 5.5 nM IC50 = 1.5 nM PMID: 10201840
RAR_beta
ZINC02007450 antagonist AGN194310 Kd = 3 +/- 2 nnM IC50 = 67 nM PMID: 10465407 
ZINC02008474 agonist Compound 5a Kd = 644 nM EC50 = 59 nM PMID: 12482435
RAR_beta
ZINC02030426 agonist Compound 3 pEC50 = 5.6 +/- 0.0 PMID: 19239230 RAR_beta
ZINC02568233 agonist TTNPB IC50 = 36 +/- 5.1 EC50 = 30 +/- 6 nM PMID: 7791761
RAR_beta
ZINC03777578 agonist Compound 13 EC50 = 740 nM PMID: 9733501
RAR_gamma
ZINC03784077 agonist AM580 Kd = 36 nM EC50 = 2 nM PMID: 12372520 RAR_gamma
ZINC03784182 agonist Compound5 Ki = 1100 +/- 70 nM AC50 = 37 +/- 7 nM PMID: 8544177 RAR_gamma
ZINC03871916 agonist Compound 1 EC50 = 13 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC03936873 agonist Compound 7 Ki = 6500 +/- 570 nM AC50 = 33 +/- 27 nM PMID: 8544177 RAR_gamma
ZINC03951146 agonist ER-34617 Relative IC50 = 2.2 +/- 1.5 Relative EC30 = 0.32 +/- 0.03 PMID: 10669568
RAR_beta
ZINC03974554 agonist Compound 12a IC50 = 9.7 Relative EC30 = 1.8 PMID: 10762039
ZINC03990465 agonist Compound 2 EC50 = 0.2 µM PMID: 16033272
ZINC04097702 agonist B-cryptoxanthin PMID: 17521617
ZINC04475360 agonist arotinoid IC50 = 36 nM EC50 = 2.1 nM PMID: 8264595
RAR_beta
ZINC04825704 agonist ALRT1550 Ki = 1.1 +/- 0.1 nM EC50 = 4.0 +/- 0.6 nM PMID: 8709094
RAR_beta
ZINC05762192 agonist Compound 4 ED30 = 54 µM Bioorg. Med. Chem. Lett. 1996 6 23 2865 RAR_beta
ZINC05762247 agonist Compound 3 Ki = 1120 +/- 200 nM AC50 = 150 +/- 21 nM PMID: 8544177
RAR_beta
ZINC06070388 agonist 3-methyl-TTNPB IC50 = 638 +/- 75 nM EC50 = 340 +/- 30 nM PMID: 8308867
RAR_beta
ZINC12358651 agonist All-trans-retinoic acid IC50 = 15 +/- 2 nM EC50 = 350 +/- 31 nM PMID: 7791761
PPAR_gamma
ZINC12661824 agonist 9-cis-retinoic acid IC50 = 7+/- 1.7 nM EC50 =191 +/- 20 nM PMID: 7791761 RAR_beta
ZINC13558478 agonist Compound 9 AC50 = 14 nM PMID: 10890153
ZINC13648516 agonist Compound 7a EC50 = 20.3 µM PMID: 16033272
ZINC13648519 agonist Compound 7b EC50 = 18.2 µM PMID: 16033272
ZINC13649044 agonist AGN 193312 Kd = 2 nM EC50 = 8 nM PMID: 12372520
RAR_beta
ZINC13649046 agonist AGN 193931 Kd = 7 nM EC50 = 94 nM PMID: 12372520
ZINC13649048 agonist AGN 194078 Kd = 3 nM EC50 = 112 nM PMID: 12372520
ZINC13652275 agonist Compound 18 EC50 = 420 nM PMID: 9733501 RAR_gamma
ZINC13652276 agonist Compound 1 EC50 = 1128 nM PMID: 10479291
ZINC13652278 agonist Compound 15 EC50 = 1000 nM PMID: 9733501
RAR_gamma
ZINC13652279 agonist Compound 17 EC50 = 2300 nM PMID: 9733501 RAR_gamma
ZINC13652284 agonist Compound 16 EC50 = 1100 nM PMID: 9733501 RAR_gamma
ZINC13676272 agonist Compound 28 PEC50 = 6.2 +/- 0.3 PMID: 19239230
RAR_beta
ZINC13734373 agonist 3-ethyl-TTNPB IC50 = 100 +/- 49 nM EC50 = 1700 +/- 118 nM PMID: 8308867
RAR_beta
ZINC13738449 agonist SR11201 EC50 = 2300 nM PMID: 7650690  RAR_beta
ZINC13742306 agonist Compound 4 EC50 = 2690 nM PMID: 7636843
RAR_beta
ZINC13742689 antagonist Compound 3 IC50 = 17 nM IC50 = 0.5 µM PMID: 7636879 RAR_gamma
ZINC13742692 antagonist Compound 26 IC50 = 14 nM IC50 = 0.36 µM PMID: 7636879 RAR_gamma
ZINC13742693 antagonist Compound 27 IC50 = 19 nM IC50 = 0.52 µM PMID: 7636879 RAR_gamma
ZINC13742694 antagonist Compound 29 IC50 = 1.2 nM IC50 = 0.21 µM PMID: 7636879 RAR_gamma
ZINC13742695 antagonist Compound 30 IC50 = 0.59 nM IC50 = 33 nM PMID: 7636879 RAR_gamma
ZINC13742696 antagonist Compound 32 IC50 = 2.3 nM IC50 = 84 nM PMID: 7636879 RAR_gamma
ZINC13742697 antagonist Compound 33 IC50 = 0.14 nM IC50 = 17 nM PMID: 7636879 RAR_gamma
ZINC13742698 antagonist Compound 34 IC50 = 16 nM IC50 = 1.3 µM PMID: 7636879 RAR_gamma
ZINC13742699 antagonist Compound 35 IC50 = 5.6 nM IC50 = 0.65 µM PMID: 7636879 RAR_gamma
ZINC13742700 antagonist Compound 36 IC50 = 3.2 nM IC50 = 0.49 µM PMID: 7636879 RAR_gamma
ZINC13742701 antagonist Compound 37 IC50 = 3.4 nM IC50 = 51 nM PMID: 7636879 RAR_gamma
ZINC13742702 antagonist Compound 38 IC50 = 4.5 nM IC50 = 0.54 µM PMID: 7636879 RAR_gamma
ZINC13742703 antagonist Compound 54 IC50 = 1.5 nM IC50 = 56 nM PMID: 7636879 RAR_gamma
ZINC13742704 antagonist Compound 39 IC50 = 19 nM IC50 = 0.1 µM PMID: 7636879 RAR_gamma
ZINC13742705 antagonist Compound 42 IC50 = 4.7 nM IC50 = 78 nM PMID: 7636879 RAR_gamma
ZINC13742706 antagonist Compound 51 IC50 = 11 nM IC50 = 77 nM PMID: 7636879 RAR_gamma
ZINC13742707 antagonist Compound 43 IC50 = 13 nM IC50 = 1.1 µM PMID: 7636879 RAR_gamma
ZINC13742708 antagonist Compound 45 IC50 = 0.97 nM IC50 = 69 nM PMID: 7636879 RAR_gamma
ZINC13742709 antagonist Compound 46 IC50 = 22 nM IC50 = 0.17 µM PMID: 7636879 RAR_gamma
ZINC13742710 antagonist Compound 47 IC50 = 3.7 nM IC50 = 37 nM PMID: 7636879 RAR_gamma
ZINC13742711 antagonist Compound 48 IC50 = 2.9 nM IC50 = 0.23 µM PMID: 7636879 RAR_gamma
ZINC13742712 antagonist Compound 49 IC50 = 30 nM IC50 = 0.3 µM PMID: 7636879
RAR_gamma
ZINC13743076 agonist SR11332 EC50 = 470 nM PMID: 7650690  RAR_beta
ZINC13743081 agonist SR11236 EC50 = 1200 NM PMID: 7650690 
RAR_gamma
ZINC13743082 agonist SR11203 EC50 = 540 nM PMID: 7650690  RAR_gamma
ZINC13743085 agonist SR11269 EC50 = 2500 nM PMID: 7650690 
RAR_beta
ZINC13745041 agonist Compound 1 Ki = 6500 +/- 2500 nM AC50 = 200 +/- 80 nM PMID: 8544177 RAR_gamma
ZINC13745049 agonist Compound 9 Ki = 695 +/- 248 nM AC50 = 7.5 +/- 4 nM PMID: 8544177 RAR_gamma
ZINC13745059 agonist Compound 12 Ki = 5000 nM AC580 = 83 +/- 28 nM PMID: 8544177
ZINC13745065 agonist Compound 14 Ki = 130 +/- 50 nM AC50 = 30 +/- 5 nM PMID: 8544177 RAR_gamma
ZINC13745067 antagonist Compound 15 Ki = 834 +/- 54 nM IC50 = 700 +/- 125 nM PMID: 8544177 RAR_gamma
ZINC13745069 agonist Compound 16 Ki = 420 +/- 110 nM AC50 = 30 +/- 16 nM PMID: 8544177 RAR_gamma
ZINC13745071 agonist Compound 17 Ki = 1056 +/- 88 nM AC50 = 300 +/- 60 nM PMID: 8544177 RAR_gamma
ZINC13745073 agonist Compound 18 Ki = 460 +/- 100 nM AC50 = 100 +/- 29 nM PMID: 8544177 RAR_gamma
ZINC13745075 agonist Compound 19 Ki = 1144 +/- 67 nM AC50 = 66 +/- 24 nM PMID: 8544177 RAR_gamma
ZINC13745077 agonist Compound 20 Ki = 610 +/- 29 nM AC50 = 1 +/- 0.41 nM PMID: 8544177
ZINC13780871 agonist Compound 10 Relative IC50 = 372 relative EC30 = 21 PMID: 9703470
RAR_beta
ZINC13781194 agonist Compound 10 EC50 = 800 nM PMID: 9733501
RAR_gamma
ZINC13781195 agonist Compound 12 EC50 = 620 nM PMID: 9733501 RAR_gamma
ZINC13781196 agonist Compound 19 EC50 = 1100 nM PMID: 9733501 RAR_gamma
ZINC13800362 agonist Compound 2 EC50 = 796 nM PMID: 10479291 RAR_gamma
ZINC13800364 agonist Compound 3 EC50 = 217 nM PMID: 10479291
ZINC13804907 agonist ER-33635 Relative IC50 = 40 +/- 2 Relative EC30 = 0.15 +/- 0.04 PMID: 10669568 RAR_beta
ZINC13804910 agonist Compound 2 Relative IC50 = 0.45 +/- 0.15 Relative EC30 = 0.34 +/- 0.1 PMID: 10669568
RAR_beta
ZINC13804918 agonist Compound 3b Relative IC50 = 32 +/- 1 ED30 = 2.1 +/- 0.4 nM PMID: 10669568 RAR_gamma
ZINC13804921 agonist Compound 3c Relative IC50 = 130 +/- 40 ED30 = 40 +/- 16 nM PMID: 10669568 RAR_gamma
ZINC13804924 agonist Compound 20c Relative IC50 = 2.4 +/- 1.4 ED30 = 9.5 +/- 3.5 nM PMID: 10669568 RAR_gamma
ZINC13804926 agonist Compound 27 b Relative IC50 = 83 +/- 9 ED30 = 11 +/- 2 nM PMID: 10669568 RAR_gamma
ZINC13809526 agonist Compound 1a Relative IC50 = 1.6 +/- 0.1 Relative EC30 = 0.8 +/- 0.14 PMID: 10956201
ZINC13809527 agonist Compound 1c Relative IC50 = 1.5 +/- 0.3 Relative EC30 = 0.7 +/- 0.15 PMID: 10956201 RAR_beta
ZINC13809529 agonist Compound 1d Relative IC50 = 15 +/- 3 Relative EC30 = 6 +/- 2.1 PMID: 10956201
ZINC13809530 agonist Compound 1e Relative IC50 = 2.5 +/- 0.3 Relative EC30 = 0.8 +/- 0.17 PMID: 10956201
ZINC13809531 agonist Compound 1g Relative IC50 = 16 +/- 3 Relative EC30 = 1.0 +/- 0.4 PMID: 10956201
ZINC13809532 agonist Compound 1h Relative IC50 = 9.4 +/- 5.0 Relative EC30 = 2.0 +/- 0.5 PMID: 10956201
ZINC13809533 agonist Compound 1i Relative IC50 = 12 +/- 8 Relative EC30 = 3.1 +/- 1.1 PMID: 10956201
ZINC13809534 agonist Compound 1j Relative IC50 = 6.1 +/- 0.4 Relative EC30 = 1.3 +/- 0.6 PMID: 10956201
ZINC13809535 agonist Compound 1k Relative IC50 = 62 +/- 21 Relative EC30 = 2.4 +/- 0.5 PMID: 10956201
ZINC13815342 agonist Compound 36 EC50 = 25 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC13815366 agonist Compound 2 Ki = 58 nM AC50 = 58 nM Bioorg. Med. Chem. Lett.1997, 7,17,2289 RAR_gamma
ZINC13815373 agonist Compound 7 Ki = 300 nM AC50 = 300 nM Bioorg. Med. Chem. Lett.1997, 7,17,2289 RAR_gamma
ZINC13815446 agonist Compound 2 EC50 = 2 µM PMID: 11405897
ZINC13815519 agonist Compound 6 Ki = 305 nM AC50 = 305 nM Bioorg. Med. Chem. Lett.1997, 7,17,2289
ZINC13815522 agonist Compound 4 Ki = 107 nM AC50 = 107 nM Bioorg. Med. Chem. Lett.1997, 7,17,2289 RAR_gamma
ZINC13832717 agonist Compound 4 EC50 = 27 nM PMID: 8410972 RAR_beta
ZINC13832718 agonist Compound 7 EC50 = 37 nM PMID: 8410972 RAR_beta
ZINC13832719 agonist Compound 8 EC50 = 45 nM PMID: 8410972 RAR_beta
ZINC13832723 agonist Compound 13 EC50 = 240 nM PMID: 8410972 RAR_beta
ZINC13832724 agonist Compound 14 EC50 = 550 nM PMID: 8410972
RAR_beta
ZINC26385838 agonist Compound 3 Ki = 34 nM AC50 = 34 nM Bioorg. Med. Chem. Lett.1997, 7,17,2289 RAR_gamma
ZINC26404528 agonist Compound 7 Kd = 52 nM EC50 = 17 nM Bioorg. Med. Chem. Lett.1997,7,18,2373
RAR_beta
ZINC26472010 agonist Compound 7 Kd = 52 nM EC50 = 17 nM Bioorg. Med. Chem. Lett.1997,7,18,2373
RAR_beta
ZINC26475061 agonist Compound 1 Kd = 5202 nM EC50 = 2300 nM Bioorg. Med. Chem. Lett.1997,7,18,2373
RAR_beta
ZINC26653776 agonist Compound 5 EC50 = 690 nM Bioorg. Med. Chem. Lett.1995,5,22,2729
RAR_beta
ZINC26657237 agonist Compound 7 EC50 = 210 nM Bioorg. Med. Chem. Lett.1995,5,22,2729 RAR_beta
ZINC26721478 agonist Compound 8 EC50 = 8 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC26723573 agonist Compound 3 EC50 = 100 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC26723692 agonist CD666 Kd = 2240 nM AC50 = 149 nM PMID: 1323296
RAR_beta
ZINC26725973 agonist Compound 5 EC50 = 25 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC26726186 agonist Compound 39 EC50 = 38 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC26726205 agonist Compound 38 EC50 = 1.3 Bioorg. Med. Chem. Lett. 1996 6 23 2865 RAR_beta
ZINC26728419 agonist Compound 6 EC50 = 25 Bioorg. Med. Chem. Lett. 1996 6 23 2865 RAR_beta
ZINC26730594 agonist Compound 10 ED30 = 92 µM Bioorg. Med. Chem. Lett. 1996 6 23 2865 RAR_beta
ZINC26731821 agonist Compound 7 EC50 = 25 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC26731825 agonist Compound 9 EC50 = 10 Bioorg. Med. Chem. Lett. 1996 6 23 2865
RAR_beta
ZINC26850547 agonist Compound 2 IC50 = 19 nM ED1/3 = 90 nM PMID: 7636879
RAR_gamma
ZINC27638789 antagonist Compound 19 Kd = 60 +/- 28 nM PMID: 10098666 RAR_beta
ZINC27645098 antagonist Compound 18 Kd = 229 +/- 48 nM PMID: 10098666 RAR_beta
ZINC27645104 antagonist Compound 17 Kd = 919 +/- 250 nM PMID: 10098666 RAR_beta
ZINC27646410 antagonist Compound 14 Kd = 85 +/- 45 nM PMID: 10098666
RAR_beta
ZINC27646416 antagonist Compound 13 Kd = 178 +/- 81 nM PMID: 10098666
RAR_beta
ZINC27647311 antagonist Compound 8 Kd = 103 +/- 17 nM PMID: 10098666
RAR_beta
ZINC27647825 antagonist Compound 7 Kd = 147 +/- 27 nM PMID: 10098666
RAR_beta
ZINC27648652 antagonist Compound 16 Kd = 44 +/- 7 nM PMID: 10098666
RAR_beta
ZINC27648730 antagonist Compound 20 Kd = 38 +/- 5 nM PMID: 10098666 RAR_beta
ZINC27650406 antagonist Compound 15 Kd = 58 +/- 9 nM PMID: 10098666 RAR_beta
ZINC27651543 antagonist Compound 9 Kd = 267 +/- 175 nM PMID: 10098666 RAR_beta
ZINC27652518 antagonist Compound 12 Kd = 90 +/- 10 nM PMID: 10098666
RAR_beta
ZINC27652522 antagonist Compound 11 Kd = 40 +/- 16 nM PMID: 10098666
RAR_beta
ZINC27652526 antagonist Compound 10 Kd = 1051 +/- 802 nM PMID: 10098666
RAR_beta
ZINC27708371 agonist Compound 1 IC50 = 2.7 Relative EC30 = 20 PMID: 10762039 RAR_beta
ZINC27710262 agonist Compound 11b IC50 = 15 Relative EC30 = 49 PMID: 10762039
ZINC27710632 agonist Compound 11a Relative IC50 = 98 Relative EC30 = 1.0 +/- 0.4 PMID: 10762038
ZINC27713389 agonist Compound 12b IC50 = 50 Relative EC30 = 4.5 PMID: 10762039
ZINC27718750 agonist Compound 11f IC50 < 1.0 Relative EC30 = 1.1 PMID: 10762039
ZINC27719619 agonist Compound 2 IC50 = 0.49 Relative EC30 = 0.27 PMID: 10762039 RAR_beta
ZINC27720272 agonist Compound 11c Relative IC50 = 7.6 Relative EC30 =0.22 PMID: 10762038
RAR_beta
ZINC27847873 antagonist Compound 2a Kd = 14 nM IC50 = 5.5 nM PMID: 10201840
RAR_beta
ZINC27858089 antagonist Compound 1a Kd  = 13 nM IC50 = 20 nM PMID: 10201840
RAR_beta
ZINC27866591 antagonist Compound 1b Kd = 15 nM IC50 = 20 nM PMID: 10201840
RAR_beta
ZINC28227159 agonist Compound 12b Relative IC50 = 1.3 ED30 = 100 nM PMID: 11354380
RAR_beta
ZINC28227625 agonist Compound 12d Relative IC50 = 1.7 ED30 = 100 nM PMID: 11354380 RAR_beta
ZINC28227633 antagonist Compound 12e Relative IC50 = 0.7 IC50 = 17 nM PMID: 11354380 RAR_beta
ZINC28227698 agonist Compound 12a Relative IC50 =5.7 ED30 = 2500 nM PMID: 11354380 RAR_beta
ZINC28227892 antagonist Compound 12c Relative IC50 = 0.8 IC50 = 1.6 nM PMID: 11354380
RAR_beta
ZINC28228318 antagonist Compound 12f Relative IC50 = 1.8 IC50 = 6.4 nM PMID: 11354380
RAR_beta
ZINC28463728 agonist Compound 8b EC50 = 6.4 µM PMID: 16033272
ZINC28758554 agonist Compound 3 AC50 = 1.0 nM PMID: 10890153
RAR_beta
ZINC28760010 agonist Compound 4 AC50 = 79 nM PMID: 10890153 RXR_alpha
ZINC28760509 agonist Compound 6 AC50 = 370 nM PMID: 10890153 RAR_beta
ZINC33973452 antagonist Compound 7 PMID: 18702457
ZINC34008167 agonist BMS753 Ki = 2 nM PMID: 10421757
ZINC38493164 agonist Compound 9 EC50 = 0.6 nM PMID: 19058965
RAR_beta
ZINC40392355 antagonist Compound 24 PMID: 18702457
ZINC40411361 antagonist Compound 11h PMID: 18702457
ZINC40897866 agonist Compound 18 pEC50 = 5.8 PMID: 19239230 RAR_beta
ZINC42891672 agonist Compound 8 pEC50 = 5.7 PMID: 19239230
RAR_beta
ZINC65731563 agonist AGN193836 Kd = 4 nM EC50 = 290 nM PMID: 12372520 RAR_beta