Compound ID Pharmacological profile Compound name Binding data Activity data Bibliographic ref Cross-reactivity
CHEMBL1080366 agonist Compound 40e EC50 = 1.87 µM PMID: 19928766
CHEMBL1081207 agonist Compound 40o EC50 = 0.46 µM PMID: 19928766
CHEMBL1081730 agonist Compound 35i EC50 = 0.018 µM PMID: 19928766
CHEMBL116540 agonist Compound 68 EC50 = 0.90 µM PMID: 12904063 PPAR_alpha
CHEMBL1169827 agonist Compound 1f EC50 = 0.9 nM PMID: 21074432
CHEMBL117402 agonist Compound 17 EC50 = 2.63 µM PMID: 15177462
PPAR_alpha
CHEMBL118577 agonist Compound 19 EC50 = 3.09 µM PMID: 15177462
PPAR_alpha
CHEMBL118816 agonist Compound 21 EC50 = 3.62 µM PMID: 15177462
PPAR_alpha
CHEMBL118939 agonist Compound 17 EC50 = 130 nM PMID: 16275077
PPAR_alpha
CHEMBL118976 agonist Compound 64 EC50 = 8.0 µM PMID: 12904063 PPAR_alpha
CHEMBL119795 agonist Compound 11 EC50 = 2.45 µM PMID: 15177462 PPAR_gamma
CHEMBL120009 agonist Compound 10 EC50 = 3.6 µM PMID: 12904063
PPAR_alpha
CHEMBL120456 agonist Compound 9 EC50 = 2.8 µM PMID: 12904063
CHEMBL120611 agonist Compound 19 EC50 = 1.5 µM PMID: 12904063 PPAR_alpha
CHEMBL120676 agonist Compound 71 EC50 = 6.60 µM PMID: 12904063 PPAR_alpha
CHEMBL120744 agonist Compound 16 EC50 = 3.0 µM PMID: 12904063
PPAR_alpha
CHEMBL120748 agonist Compound 57 EC50 = 0.40 µM PMID: 12904063
CHEMBL122070 agonist Compound 74 EC50 = 3.0 µM PMID: 12904063
PPAR_alpha
CHEMBL1222408 agonist Compound 11d EC50 = 120 +/- 10 nM PMID: 21530275 PPAR_alpha
CHEMBL1630380 agonist Compound 1i EC50 = 4.5 nM PMID: 21074432
PPAR_alpha
CHEMBL1630381 agonist Compound 1h EC50 = 6.2 nM PMID: 21074432 PPAR_alpha
CHEMBL1630382 agonist Compound 1g EC50 = 11.0 nM PMID: 21074432 PPAR_alpha
CHEMBL1630383 agonist Compound 2f EC50 = 1.0 nM PMID: 21074432 PPAR_alpha
CHEMBL1630384 agonist Compound 2i EC50 = 1.8 nM PMID: 21074432
PPAR_alpha
CHEMBL1630385 agonist Compound 2h EC50 = 7.0 nM PMID: 21074432 PPAR_gamma
CHEMBL1630386 agonist Compound 2g EC50 = 8.5 nM PMID: 21074432
CHEMBL1634195 agonist Compound 10 EC50 = 0.32 µM PMID: 21094606
CHEMBL1643192 agonist Compound 3 EC50 = 1.6 µM PMID: 21094606
CHEMBL1643193 agonist Compound 4 EC50 = 1.0 µM PMID: 21094606
CHEMBL1643194 agonist Compound 5 EC50 = 0.025 µM PMID: 21094606
CHEMBL1643196 agonist Compound 11 EC50 = 2.5 µM PMID: 21094606
CHEMBL1643202 agonist Compound 20 EC50 = 0.5 µM PMID: 21094606
CHEMBL1643203 agonist Compound 21 EC50 = 2.0 µM PMID: 21094606
CHEMBL1760269 agonist Compound 13 pIC50 = 7.2 PEC50 = 6.9 PMID: 21414782
CHEMBL1760274 agonist Compound 16 pIC50 = 7.8 PEC50 = 7.8 PMID: 21414782
CHEMBL1760399 agonist Compound 17 pIC50 = 7.1 PEC50 = 7.2 PMID: 21414782
CHEMBL1760400 agonist Compound 18 pIC50 = 6.8 PEC50 = 6.5 PMID: 21414782
CHEMBL1760401 agonist Compound 19 pIC50 = 6.6 PEC50 = 6.4 PMID: 21414782
CHEMBL1760402 agonist Compound 20 pIC50 = 6.3 PEC50 = 6.3 PMID: 21414782
CHEMBL1760403 agonist Compound 21 pIC50 = 6.2 PEC50 = 6.5 PMID: 21414782
CHEMBL1760405 agonist Compound 23 pIC50 = 6.9 PEC50 = 7.1 PMID: 21414782
CHEMBL1760406 agonist Compound 24 pIC50 = 6.1 PEC50 = 6.4 PMID: 21414782
CHEMBL1760407 agonist Compound 25 pIC50 = 6.0 PEC50 = 6.3 PMID: 21414782
CHEMBL1760408 agonist Compound 26 pIC50 = 6.1 PEC50 = 6.1 PMID: 21414782
CHEMBL1760409 agonist Compound 27 pIC50 = 6.3 PEC50 = 6.3 PMID: 21414782
CHEMBL1760410 agonist Compound 28 pIC50 = 5.9 PEC50 = 5.7 PMID: 21414782
CHEMBL1779473 agonist Compound 11c EC50 = 110 +/- 12 nM PMID: 21530275 PPAR_alpha
CHEMBL1779474 agonist Compound 11e EC50 = 4800 +/- 700 nM PMID: 21530275 PPAR_alpha
CHEMBL1779476 agonist Compound 11h EC50 = 4100 +/- 400 nM PMID: 21530275 PPAR_alpha
CHEMBL1779478 agonist Compound 11j EC50 = 1400 +/- 300 nM PMID: 21530275 PPAR_alpha
CHEMBL1779479 agonist Compound 11k EC50 = 1400 +/- 100 nM PMID: 21530275 PPAR_alpha
CHEMBL1813188 agonist Compound 11a EC50 = 13 µM PMID: 21514830
PPAR_alpha
CHEMBL1813191 agonist Compound 12a EC50 = 29 µM PMID: 21514830 PPAR_alpha
CHEMBL1813194 agonist Compound 13a EC50 = 14 µM PMID: 21514830
PPAR_alpha
CHEMBL1813195 agonist Compound 13b EC50 = 25 µM PMID: 21514830
PPAR_alpha
CHEMBL1813199 agonist Compound 13f EC50 = 3.2 µM PMID: 21514830
PPAR_alpha
CHEMBL1813200 agonist Compound (S) 13c EC50 = 7.3 µM PMID: 21514830 PPAR_gamma
CHEMBL1813202 agonist Compound (S) 13d EC50 = 1.9 µM PMID: 21514830 PPAR_gamma
CHEMBL1813203 agonist Compound (R) 13d EC50 = 9.7 µM PMID: 21514830 PPAR_gamma
CHEMBL1813204 agonist Compound (S) 13e EC50 = 1.8 µM PMID: 21514830 PPAR_gamma
CHEMBL1927473 agonist Compound 2a EC50 = 55 +/- 4 nM PMID: 22051054 PPAR_alpha
CHEMBL1927474 agonist Compound 2b EC50 = 290 +/- 12 nM PMID: 22051054 PPAR_alpha
CHEMBL1927475 agonist Compound 2c EC50 = 580 +/- 28 nM PMID: 22051054 PPAR_alpha
CHEMBL1934480 agonist Compound 14c EC50 = 7.1 µM PMID: 22133631
CHEMBL1934481 agonist Compound 14d EC50 = 2.4 µM PMID: 22133631 PPAR_alpha
CHEMBL1934482 agonist Compound 14e EC50 = 1.9 µM PMID: 22133631 PPAR_alpha
CHEMBL1934483 agonist Compound 14f EC50 = 8.8 µM PMID: 22133631 PPAR_alpha
CHEMBL1934484 agonist Compound 14g EC50 = 3.1 µM PMID: 22133631 PPAR_alpha
CHEMBL1934485 agonist Compound 14h EC50 = 43 nM PMID: 22133631 PPAR_alpha
CHEMBL200495 agonist Compound 5 IC50 = 0.096 EC50 = 0.010 µM PMID: 16451087
PPAR_alpha
CHEMBL2011544 agonist Compound 11 EC50 = 4.9 +/- 0.7 µM PMID: 22381047 PPAR_gamma
CHEMBL201581 agonist Compound 10c IC50 = 3.153 µM EC50 = 4.350 µM PMID: 16451087 PPAR_alpha
CHEMBL201653 agonist Compound 10d IC50 = 3.256 µM EC50 = 4.000 µM PMID: 16451087 PPAR_alpha
CHEMBL201803 agonist Compound 10c EC50 = 500 nM PMID: 16275077
PPAR_alpha
CHEMBL201832 agonist Compound 10b EC50 = 1000 nM PMID: 16275077
PPAR_alpha
CHEMBL201880 agonist Compound 10k IC50 = 0.223 µM EC50 = 0.500 µM PMID: 16451087
PPAR_alpha
CHEMBL202140 agonist Compound 10f IC50 = 7.616 µM EC50 = 5.290 µM PMID: 16451087 PPAR_gamma
CHEMBL202246 agonist Compound 10l IC50 = 2.398 µM EC50 = 4.900 µM PMID: 16451087
PPAR_alpha
CHEMBL202617 agonist Compound 10h IC50 = 4.430 µM EC50 = 5.600 µM PMID: 16451087
PPAR_alpha
CHEMBL2035057 agonist Compound 11t EC50 = 1.1 nM PMID: 22534184
CHEMBL2035058 agonist Compound 11f EC50 = 1.2 nM PMID: 22534184
CHEMBL2035059 agonist Compound 11g EC50 = 2.8 nM PMID: 22534184
CHEMBL2035060 agonist Compound 11h EC50 = 4.6 nM PMID: 22534184
CHEMBL2035061 agonist Compound 11i EC50 = 16.7 nM PMID: 22534184
CHEMBL2035062 agonist Compound 11j EC50 = 6.7 nM PMID: 22534184
CHEMBL2035063 agonist Compound 11k EC50 = 8.1 nM PMID: 22534184
CHEMBL2035064 agonist Compound 11l EC50 = 4.4 nM PMID: 22534184
CHEMBL2035065 agonist Compound 11m EC50 = 490.1 nM PMID: 22534184
CHEMBL2035067 agonist Compound 11o EC50 = 523.0 nM PMID: 22534184
CHEMBL2035068 agonist Compound 11p EC50 = 1.8 nM PMID: 22534184
CHEMBL2035069 agonist Compound 11q EC50 = 1.0 nM PMID: 22534184
CHEMBL2035070 agonist Compound 11r EC50 = 2.3 nM PMID: 22534184
CHEMBL2035071 agonist Compound 11s EC50 = 1.1 nM PMID: 22534184
CHEMBL2037577 agonist Compound 10a EC50 = 1.6 nM PMID: 22534184
CHEMBL2037578 agonist Compound 10b EC50 = 2.6 nM PMID: 22534184
CHEMBL2037579 agonist Compound 10c EC50 = 6.1 nM PMID: 22534184
CHEMBL2037580 agonist Compound 10d EC50 = 38.8 nM PMID: 22534184
CHEMBL2037581 agonist Compound 10e EC50 = 11.4 nM PMID: 22534184
CHEMBL2037582 agonist Compound 10f EC50 = 57.2 nM PMID: 22534184
CHEMBL2037583 agonist Compound 10g EC50 = 132 nM PMID: 22534184
CHEMBL2037584 agonist Compound 11a EC50 = 60.0 nM PMID: 22534184
CHEMBL2037585 agonist Compound 11b EC50 = 9.4 nM PMID: 22534184
CHEMBL2037586 agonist Compound 11c EC50 = 4.8 nM PMID: 22534184
CHEMBL2037587 agonist Compound 11d EC50 = 1.2 nM PMID: 22534184
CHEMBL2037588 agonist Compound 11e EC50 = 2.1 nM PMID: 22534184
CHEMBL2064743 agonist MDG582 EC50 = 26.0 +/- 3.6 µM PMID: 22582973 PPAR_gamma
CHEMBL212023 agonist Compound 12 IC50 = 9 +/- 0 nM EC50 = 52 +/- 12 nM PMID: 16970391 PPAR_gamma
CHEMBL215127 agonist Compound 11 IC50 = 6 +/- 1 nM EC50 = 25 +/- 5 nM PMID: 16970391
PPAR_alpha
CHEMBL215582 agonist Compound 7 IC50 = 5 +/- 0 nM EC50 = 45 +/- 8 nM PMID: 16970391
PPAR_alpha
CHEMBL229525 agonist Compound 10f EC50 = 5.1 +/- 0.5 nM PMID: 17532641
PPAR_alpha
CHEMBL229573 agonist Compound 10g EC50 = 1.8 +/- 0.3 nM PMID: 17532641
PPAR_alpha
CHEMBL229778 agonist Compound 5c EC50 = 6.8 +/- 0.6 nM PMID: 17532641
PPAR_alpha
CHEMBL229785 agonist Compound 10b EC50 = 120 +/- 10 nM PMID: 17532641 PPAR_alpha
CHEMBL229786 agonist Compound 10c EC50 = 700 +/- 150 nM PMID: 17532641
PPAR_alpha
CHEMBL229831 agonist Compound 5e EC50 = 45 +/- 5 nM PMID: 17532641
PPAR_alpha
CHEMBL229837 agonist Compound 10e EC50 = 220 +/- 20 nM PMID: 17532641
PPAR_alpha
CHEMBL229888 agonist Compound 10a EC50 = 210 +/- 30 nM PMID: 17532641 PPAR_alpha
CHEMBL230177 agonist Compound 16 EC50 = 6.9 nM PMID: 17524639
CHEMBL230179 agonist Compound 18 EC50 = 24.3 nM PMID: 17524639
CHEMBL230268 agonist Compound 5 EC50 = 7.0 nM PMID: 17524639
CHEMBL230269 agonist Compound 6 EC50 = 3.9 nM PMID: 17524639
CHEMBL230372 agonist Compound 2 EC50 = 18.8 nM PMID: 17524639
CHEMBL230605 agonist Compound 8 EC50 = 60.0 nM PMID: 17524639
CHEMBL231527 agonist Compound 11 EC50 = 23.9 nM PMID: 17524639
CHEMBL231528 agonist Compound 12 EC50 = 4.6 nM PMID: 17524639
CHEMBL231531 agonist Compound 13 EC50 = 17.0 nM PMID: 17524639
CHEMBL231696 agonist Compound 6b EC50 = 0.011 µM PMID: 17553681
CHEMBL234485 agonist Compound 6d EC50 = 0.77 µM PMID: 17553681
CHEMBL234689 agonist Compound 6e EC50 = 0.24 µM PMID: 17553681
CHEMBL234691 agonist Compound 6j EC50 = 0.49 µM PMID: 17553681
CHEMBL234692 agonist Compound 6k EC50 = 3.0 µM PMID: 17553681
CHEMBL234693 agonist Compound 6m EC50 = 1.2 µM PMID: 17553681
CHEMBL234903 agonist Compound 6f EC50 = 0.13 µM PMID: 17553681
CHEMBL234904 agonist Compound 6g EC50 = 0.32 µM PMID: 17553681
CHEMBL234905 agonist Compound 6h EC50 = 2.0 µM PMID: 17553681
CHEMBL234906 agonist Compound 6n EC50 = 3.9 µM PMID: 17553681
CHEMBL234907 agonist Compound 6o EC50 = 0.15 µM PMID: 17553681 PPAR_alpha
CHEMBL234908 agonist Compound 6q EC50 = 0.29 µM PMID: 17553681
PPAR_alpha
CHEMBL239351 agonist Compound 10 EC50 = 24 nM PMID: 17157013 PPAR_alpha
CHEMBL245464 agonist Compound 30 EC50 = 0.16 µM PMID: 17553678
PPAR_alpha
CHEMBL245465 agonist Compound 31 EC50 = 5.0 µM PMID: 17553678 PPAR_alpha
CHEMBL245664 agonist Compound 34 EC50 = 0.14 µM PMID: 17553678 PPAR_alpha
CHEMBL246069 agonist Compound 38 EC50 = 1.4 µM PMID: 17553678 PPAR_alpha
CHEMBL246070 agonist Compound 40 EC50 = 0.12 µM PMID: 17553678
PPAR_alpha
CHEMBL246281 agonist Compound 42 EC50 = 0.83 µM PMID: 17553678
PPAR_alpha
CHEMBL246282 agonist Compound 43 EC50 = 6.5 µM PMID: 17553678 PPAR_gamma
CHEMBL246510 agonist Compound 45 EC50 = 0.003 µM PMID: 17553678
PPAR_alpha
CHEMBL248324 agonist Compound 23 EC50 = 2.7 µM PMID: 17553678
PPAR_alpha
CHEMBL248326 agonist Compound 25 EC50 = 2.3 µM PMID: 17553678
PPAR_alpha
CHEMBL248526 agonist Compound 26 EC50 = 1.4 µM PMID: 17553678
PPAR_alpha
CHEMBL248527 agonist Compound 28 EC50 = 1.9 µM PMID: 17553678
PPAR_alpha
CHEMBL255392 agonist Compound 11b EC50 = 360 +/- 40 nM PMID: 21530275
PPAR_alpha
CHEMBL255426 agonist Compound 10l EC50 = 810 nM PMID: 18162399
PPAR_alpha
CHEMBL255593 agonist Compound 11a EC50 = 8100 +/- 400 nM PMID: 21530275 PPAR_alpha
CHEMBL262558 agonist Compound 52 EC50 = 0.64 µM PMID: 12904063
CHEMBL270451 agonist Compound 10i EC50 = 1400 nM PMID: 18162399
PPAR_alpha
CHEMBL270587 agonist Compound 11g EC50 = 210 +/- 20 nM PMID: 21530275
PPAR_alpha
CHEMBL270664 agonist Compound 10j EC50 = 250 nM PMID: 18162399
PPAR_alpha
CHEMBL270801 agonist Compound 10e EC50 = 300 nM PMID: 18162399
PPAR_alpha
CHEMBL271877 agonist Compound 10c EC50 = 720 nM PMID: 18162399
PPAR_alpha
CHEMBL305723 agonist Compound 2b EC50 = 4000 nM PMID: 11527737
PPAR_alpha
CHEMBL307728 agonist Compound 1n EC50 = 320 nM PMID: 11527737
PPAR_alpha
CHEMBL309778 agonist Compound 1m EC50 = 160 nM PMID: 11527737
PPAR_alpha
CHEMBL310426 agonist Compound 1f EC50 = 2500 nM PMID: 11527737
PPAR_alpha
CHEMBL310962 agonist Compound 1h EC50 = 790 nM PMID: 11527737
PPAR_alpha
CHEMBL311429 agonist Compound 1a EC50 = 10000 nM PMID: 11527737
PPAR_alpha
CHEMBL312791 agonist Compound 1i EC50 = 500 nM PMID: 11527737
PPAR_alpha
CHEMBL325723 agonist Compound 27 EC50 = 3.0 µM PMID: 12904063
PPAR_alpha
CHEMBL33188 agonist Compound 16 EC50 = 1.05 µM PMID: 15177462
PPAR_alpha
CHEMBL332465 agonist Compound 11 EC50 = 2.4 µM PMID: 12904063 PPAR_alpha
CHEMBL376165 agonist Compound 5h EC50 = 1.7 +/- 0.1 nM PMID: 17532641
PPAR_alpha
CHEMBL387914 agonist Compound 5g EC50 = 21 +/- 1 nM PMID: 17532641
PPAR_alpha
CHEMBL389769 agonist Compound 4 EC50 = 4.3 nM PMID: 17524639
CHEMBL389903 agonist Compound 5d EC50 = 4.8 +/- 0.6 nM PMID: 17532641
PPAR_alpha
CHEMBL390004 agonist Compound 14 EC50 = 7.4 nM PMID: 17524639
CHEMBL390116 agonist Compound 10d EC50 = 40 +/- 6 nM PMID: 17532641
PPAR_alpha
CHEMBL390199 agonist Compound 17 EC50 = 15.2 nM PMID: 17524639
CHEMBL391620 agonist Compound 44 EC50 = 1.3 µM PMID: 17553678
PPAR_alpha
CHEMBL392810 agonist Compound 33 EC50 = 1.9 µM PMID: 17553678
PPAR_alpha
CHEMBL393186 agonist Compound 6a EC50 = 0.16 µM PMID: 17553681
CHEMBL393987 agonist Compound 6i EC50 = 0.22 µM PMID: 17553681
CHEMBL397218 agonist Compound 9 EC50 = 126 nM PMID: 17524639
CHEMBL397449 agonist Compound 10 EC50 = 62.1 nM PMID: 17524639
CHEMBL397970 agonist Compound 1 EC50 = 79.0 nM PMID: 17524639
CHEMBL398117 agonist Compound 27 EC50 = 1.1 µM PMID: 17553678
PPAR_alpha
CHEMBL398118 agonist Compound 29 EC50 = 8.0 µM PMID: 17553678
PPAR_alpha
CHEMBL402161 agonist Compound 4e EC50 = 940 +/- 30 nM PMID: 18662876
PPAR_alpha
CHEMBL425666 agonist Compound 5b EC50 = 15 +/- 4 nM PMID: 17532641 PPAR_gamma
CHEMBL425766 agonist Compound 10e IC50 = 0.649 µM EC50 = 0.610 µM PMID: 16451087
PPAR_alpha
CHEMBL426371 agonist Compound 5f EC50 = 110 +/- 20 nM PMID: 17532641 PPAR_gamma
CHEMBL426483 agonist Compound  18 EC50 = 2000 nM PMID: 16275077 PPAR_alpha
CHEMBL427701 agonist Compound 41 EC50 = 0.11 µM PMID: 17553678
PPAR_alpha
CHEMBL428574 agonist Compound 32 EC50 = 1.1 µM PMID: 17553678
PPAR_alpha
CHEMBL429824 agonist Compound 37 EC50 = 1.7 µM PMID: 17553678
PPAR_alpha
CHEMBL433306 agonist Compound 1d EC50 = 1600 nM PMID: 11527737
PPAR_alpha
CHEMBL433316 agonist Compound 2g EC50 = 2500 nM PMID: 11527737
PPAR_alpha
CHEMBL437364 agonist Compound 6p EC50 = 0.29 µM PMID: 17553681
CHEMBL455957 agonist Compound 4c EC50 = 59 +/- 6 nM PMID: 18662876 PPAR_alpha
CHEMBL456752 agonist Compound 4f EC50 = 550 +/- 70 nM PMID: 18662876
PPAR_alpha
CHEMBL456753 agonist Compound 4g EC50 = 2200 +/- 300 nM PMID: 18662876
PPAR_alpha
CHEMBL456973 agonist Compound 4h EC50 = 280 +/- 30 nM PMID: 18662876
PPAR_alpha
CHEMBL456974 agonist Compound 4i EC50 = 94 +/- 9 nM PMID: 18662876
PPAR_alpha
CHEMBL457405 agonist Compound 4k EC50 = 55 +/- 3 nM PMID: 18662876
PPAR_alpha
CHEMBL462982 agonist Compound 4d EC50 = 20 +/- 2 nM PMID: 18662876
PPAR_alpha
CHEMBL501980 agonist Compound 16 Ki = 0.070 µM EC50 = 7.1 µM PMID: 19464171
CHEMBL508953 agonist Compound 7f Transactivation = 1.8 PMID: 18805005 PPAR_gamma
CHEMBL514256 agonist Compound 4j EC50 = 60 +/- 7 nM PMID: 18662876
PPAR_alpha
CHEMBL76676 agonist Compound 1l EC50 = 5000 nM PMID: 11527737
PPAR_alpha
CHEMBL78442 agonist Compound 2e EC50 = 100 nM PMID: 11527737
PPAR_alpha
CHEMBL78523 agonist Compound 1c EC50 = 7900 nM PMID: 11527737
PPAR_alpha
CHEMBL80301 agonist Compound 1e EC50 = 1600 nM PMID: 11527737
PPAR_alpha
CHEMBL80364 agonist Compound 1k EC50 = 7900 nM PMID: 11527737
PPAR_alpha
CHEMBL80671 agonist Compound 1g EC50 = 500 nM PMID: 11527737
PPAR_alpha
CHEMBL80772 agonist Compound 1b EC50 = 7900 nM PMID: 11527737
PPAR_alpha
CHEMBL80791 agonist Compound 2f EC50 = 500 nM PMID: 11527737
PPAR_alpha
CHEMBL80905 agonist Compound 1j EC50 = 7900 nM PMID: 11527737
PPAR_alpha
ZINC00388674 agonist Compound 9 EC50 = 50.6 +/- 5.3 µM PMID: 22381047 PPAR_gamma
ZINC00593304 agonist Compound 3 EC50 = 14.9 µM PMID: 21515063
PPAR_alpha
ZINC00593306 agonist Compound 7 EC50 = 6.7 µM PMID: 21515063
PPAR_alpha
ZINC00593307 agonist Compound 8 EC50 = 9.8 µM PMID: 21515063
PPAR_alpha
ZINC00603089 agonist Compound 9 EC50 = 5.4 µM PMID: 21515063
PPAR_alpha
ZINC01549535 agonist Compound 20 EC50 = 1.0 µM PMID: 12482434
PPAR_alpha
ZINC01549989 agonist gw501516 IC50 = 1 +/- 0.1 nM EC50 = 0.85 +/- 0.29 µM PMID: 12699745
ZINC01553970 agonist Compound 19 EC50 = 0.5 µM PMID: 12482434
PPAR_alpha
ZINC01553971 agonist Compound 1 EC50 = 0.54 +/- 0.05 µM PMID: 17343371
PPAR_alpha
ZINC01554219 agonist Compound 9 Ki = 0.3 nM EC50 = 20 nM PMID: 12617924
PPAR_alpha
ZINC01554220 agonist Compound 6 Ki = 93 nM max at 3 µM = 86% PMID: 12617924
PPAR_alpha
ZINC01554391 agonist L-796449 IC50 = 6 nM EC50 = 6 nM PMID: 12657263
PPAR_alpha
ZINC02541693 agonist L-165041 EC50 = 125 nM PMID: 16797985
PPAR_alpha
ZINC03817280 agonist Compound 10a IC50 = 3.1 nM EC50 = 14.7 nM PMID: 17512197
ZINC03819472 agonist NNC 61-3058 EC50 = 9.6 µM PMID: 17379517 
PPAR_alpha
ZINC03819473 agonist Compound 6 EC50 = 6.90 +/- 1.08 µM PMID: 14584939
PPAR_alpha
ZINC03834054 agonist L-783483 IC50 = 10 nnM EC50 = 5 nM PMID: 12657263
LXR_alpha
ZINC03870758 agonist gw2433 EC50 = 0.19 µM PMID: 10691680
ZINC03940632 agonist Compound 4e Ki = 2500 nM EC50 = 3800 nM PMID: 11720854
PPAR_alpha
ZINC03949277 agonist Compound 8 EC50 = 0.017 +/- 0.001 µM PMID: 17343371
ZINC03949282 agonist Compound 7 EC50 = 0.053 +/- 0.003 µM PMID: 17343371
ZINC03961820 agonist Compound 13 EC50 = 34 nM PMID: 17157013
ZINC03961821 agonist Compound 34v EC50 = 18 nM PMID: 17274610 PPAR_alpha
ZINC03961822 agonist Compound 34z EC50 = 218 nM PMID: 17274610
ZINC03961823 agonist Compound 34ak EC50 = 3 nM PMID: 17274610 PPAR_alpha
ZINC03961825 agonist Compound 34ad EC50 = 4.6 nM PMID: 17274610 PPAR_alpha
ZINC03961827 agonist Compound 34t EC50 = 5.2 nM PMID: 17274610 PPAR_alpha
ZINC03976748 agonist Compound 10 EC50 = 0.004 µM PMID: 17243659 PPAR_gamma
ZINC04777896 agonist Compound 3 EC50 = 49.5 +/- 4.8 µM PMID: 22381047 PPAR_gamma
ZINC06001877 agonist Compound 6 EC50 = 33.9 +/- 3.6 µM PMID: 22381047 PPAR_gamma
ZINC08022594 agonist gw0742 IC50 = 1 +/- 0.01 nM EC50 = 1 +/- 0.2 nM PMID: 12699745 PPAR_gamma
ZINC08455242 agonist MDG559 EC50 = 21.0 +/- 6.7 µM PMID: 22582973 PPAR_gamma
ZINC09933928 antagonist Compound 9 IC50 = 7.2 µM PMID: 18821746
ZINC1024901 antagonist gsk3787 pIC50 = 6.7 pIC50 = 6.9 PMID: 20128594 
ZINC12358141 agonist Compound 4 EC50 = 0.79 µM PMID: 10508427
PPAR_alpha
ZINC12358209 agonist Compound 7 EC50 = 5.7 µM PMID: 12482434
PPAR_alpha
ZINC12358210 agonist Compound 8 EC50 = 8.3 µM PMID: 12482434
PPAR_alpha
ZINC12358211 agonist Compound 9 EC50 = 3.4 µM PMID: 12482434
PPAR_alpha
ZINC12358212 agonist Compound 10 EC50 = 2.2 µM PMID: 12482434
PPAR_alpha
ZINC12358213 agonist Compound 11 EC50 = 2.2 µM PMID: 12482434
PPAR_alpha
ZINC12358214 agonist Compound 12 EC50 = 0.9 µM PMID: 12482434
PPAR_alpha
ZINC12358215 agonist Compound 13 EC50 = 3.4 µM PMID: 12482434
PPAR_alpha
ZINC12358216 agonist Compound 14 EC50 = 0.6 µM PMID: 12482434
PPAR_alpha
ZINC12358217 agonist Compound 15 EC50 = 2.0 µM PMID: 12482434
PPAR_alpha
ZINC12358218 agonist Compound 16 EC50 = 2.0 µM PMID: 12482434
PPAR_alpha
ZINC12358219 agonist Compound 17 EC50 = 0.7 µM PMID: 12482434
PPAR_alpha
ZINC12358236 agonist Compound 2 Ki = 3.7 nM max at 3 µM = 34 % PMID: 12617924
PPAR_alpha
ZINC12358237 agonist Compound 4 Ki = 508.0 nM EC50 = 147 nM PMID: 12617924
PPAR_alpha
ZINC12358238 agonist Compound 5 Ki = 5 nM EC50 = 3 nM PMID: 12617924
PPAR_alpha
ZINC12358239 agonist Compound 7 Ki = 203 nM max at 3 µM = 59% PMID: 12617924
PPAR_alpha
ZINC12358240 agonist Compound 10 Ki = 165 nM EC50 = 400 nM PMID: 12617924
PPAR_alpha
ZINC12358241 agonist Compound 14 Ki = 2 nM Max % at 3µM = 74 % PMID: 12617924
PPAR_alpha
ZINC12358242 agonist Compound 15 Ki = 37.5 nM Max % at 3µM = 74 % PMID: 12617924
PPAR_alpha
ZINC12358243 agonist Compound 16 Ki = 529 nM Max % at 3µM = 18% PMID: 12617924
PPAR_alpha
ZINC12358244 agonist Compound 17 Ki = 317 nM EC50 = 860 nM PMID: 12617924
PPAR_alpha
ZINC12358245 agonist Compound 27 Ki = 18 nM EC50 = 148 nM PMID: 12617924
PPAR_alpha
ZINC12358246 agonist Compound 28 Ki = 265 nM EC50 = 640 nM PMID: 12617924
PPAR_alpha
ZINC12358247 agonist Compound 18 Ki = 3.7 nM EC50 = 16 nM PMID: 12617924
PPAR_alpha
ZINC12358248 agonist Compound 19 Ki = 4.6 nM EC50 = 13 nM PMID: 12617924
PPAR_alpha
ZINC12358250 agonist Compound 20 Ki = 136 nM Max % at 3µM = 117% PMID: 12617924
PPAR_alpha
ZINC12358252 agonist Compound 21 Ki = 23 nM EC50 = 172 nM PMID: 12617924
PPAR_alpha
ZINC12358253 agonist Compound 24 Ki = 47 nM Max % at 3µM = 127% PMID: 12617924
PPAR_alpha
ZINC12358254 agonist Compound 25 Ki = 110 nM Max % at 3µM = 85% PMID: 12617924
PPAR_alpha
ZINC12358255 agonist Compound 29 Ki = 156 nM Max % at 3µM = 69% PMID: 12617924
PPAR_alpha
ZINC12358256 agonist Compound 30 Ki = 38 nM EC50 = 183 nM PMID: 12617924
PPAR_alpha
ZINC12358257 agonist Compound 1 IC50 = 20 nM EC50 = 80 nM PMID: 12657263
PPAR_alpha
ZINC12358258 agonist Compound 2 IC50 = 20 nM EC50 = 10 nM PMID: 12657263
PPAR_alpha
ZINC12358259 agonist Compound 3 IC50 = 10 nM EC50 = 9 nM PMID: 12657263
PPAR_alpha
ZINC12358260 agonist L-165461 IC50 = 4 nM EC50 = 11 nM PMID: 12657263
PPAR_alpha
ZINC12358261 agonist Compound 6 IC50 = 40 nM EC50 = 12 nM PMID: 12657263
PPAR_alpha
ZINC12358348 agonist Compound 15 IC50 =1200 +/- 120 nM EC50 = 3000 +/- 19 nM PMID: 14613314
PPAR_alpha
ZINC12358350 agonist Compound 17 IC50 = 880 +/- 31 nM EC50 = 3000 +/- 20 nM PMID: 14613314
PPAR_alpha
ZINC12358351 agonist Compound 18 IC50 = 1700 +/- 15 nM EC50 = 3000 +/- 20 nM PMID: 14613314
PPAR_alpha
ZINC12358352 agonist Compound 19 IC50 = 740 +/- 70 nM EC50 = 2900 +/- 8 nM PMID: 14613314
PPAR_alpha
ZINC12504466 agonist Compound 2 EC50 = 0.500 µM PMID: 17034149
PPAR_alpha
ZINC13260173 agonist Compound 4 pIC50 = 8.1 PEC50 = 6.9 PMID: 18722772
ZINC13489471 agonist Compound 7a IC50 = 1.0 +/- 0.07 µM EC50 = 1.9 +/- 0.39 µM PMID: 12699745 PPAR_gamma
ZINC13489472 agonist Compound 7b IC50 = 0.03 +/- 0.002 µM EC50 = 0.09 +/- 0.02 µM PMID: 12699745 PPAR_gamma
ZINC13489473 agonist Compound 7c IC50 = 1.0 +/- 0.03 µM EC50 = 0.02 +/- 0.006 µM PMID: 12699745 PPAR_gamma
ZINC13489474 agonist Compound 7d IC50 = 0.06 µM EC50 = 0.03 +/- 0.03 µM PMID: 12699745 PPAR_gamma
ZINC13489475 agonist Compound 7e IC50 = 0.09 +/- 0.003 µM EC50 = 0.06 +/- 0.02 µM PMID: 12699745 PPAR_gamma
ZINC13489476 agonist Compound 7f IC50 = 5.5 +/- 0.28 µM EC50 = 5.9 +/- 5.5 µM PMID: 12699745
ZINC13489477 agonist Compound 7g IC50 = 0.34 +/- 0.008 µM EC50 = 0.47 +/- 0.18 µM PMID: 12699745 PPAR_gamma
ZINC13489478 agonist Compound 7h IC50 = 0.03 +/- 0.001 µM EC50 = 0.03 +/- 0.002 µM PMID: 12699745
ZINC13489479 agonist Compound 7i IC50 = 0.09 +/- 0.002 µM EC50 = 0.42 +/- 0.18 µM PMID: 12699745 PPAR_gamma
ZINC13489480 agonist Compound 7j IC50 = 0.001 +/- 0.0001 µM EC50 = 0.01 +/- 0.001 µM PMID: 12699745 PPAR_gamma
ZINC13980247 agonist Compound 10 IC50 = 183 +/- 0 nM EC50 = 339 +/- 0 nM PMID: 16970391 PPAR_gamma
ZINC13981352 agonist Compound 32 EC50 = 8.6 nM PMID: 19168353
ZINC13981353 agonist Compound 5 EC50 = 17.1 nM PMID: 19168353
ZINC13981355 agonist Compound 13 EC50 = 26.8 nM PMID: 19168353
ZINC13981356 agonist Compound 10 EC50 = 28.4 nM PMID: 19168353
ZINC13981358 agonist Compound 30 EC50 = 22.4 nM PMID: 19168353
ZINC13981360 agonist Compound 31 EC50 = 23.3 nM PMID: 19168353
ZINC13982030 agonist Compound 13 EC50 (%inhibition) = 42.6 PMID: 18083521
PPAR_alpha
ZINC13983071 agonist Compound 11 EC50 = 2.060 µM PMID: 18947994
PPAR_alpha
ZINC13983075 agonist Compound 9 EC50 = 4.850 µM PMID: 18947994
PPAR_alpha
ZINC13983079 agonist Compound 27 EC50 = 1.63 µM PMID: 18947994
PPAR_alpha
ZINC13983521 agonist Compound 13a Transactivation = 1.0 PMID: 18805005 PPAR_gamma
ZINC13983527 agonist Compound 9 Transactivation = 1.0 PMID: 18805005 PPAR_gamma
ZINC13985145 agonist Compound 2 EC50 = 0.003 µM PMID: 21094606
ZINC14096589 agonist Compound 5 EC50 = 3.1 µM PMID: 10508427
PPAR_alpha
ZINC14115100 agonist gw9578 EC50 = 1.4 µM PMID: 10691680
PPAR_alpha
ZINC14209392 agonist Compound 9 IC50 = 3 +/- 1 nM EC50 = 5 +/- 1 nM PMID: 16970391
PPAR_alpha
ZINC14209394 agonist Compound 14 IC50 = 4 +/- 0 nM EC50 = 5 +/- 0 nM PMID: 16970391
PPAR_alpha
ZINC14588894 agonist Compound 7 EC50 = 48.5 +/- 4.2 µM PMID: 22381047 PPAR_gamma
ZINC14976992 agonist Compound 17a EC50 = 44 nM PMID: 17274610
ZINC14976995 agonist Compound 17b EC50 = 8.9 nM PMID: 17274610 PPAR_alpha
ZINC14976998 agonist Compound 17c EC50 = 4.2 nM PMID: 17274610 PPAR_alpha
ZINC14977001 agonist Compound 17d EC50 = 13 nM PMID: 17274610 PPAR_alpha
ZINC14977004 agonist Compound 17e EC50 = 6.7 nM PMID: 17274610
ZINC14977007 agonist Compound 17f EC50 = 6.6 nM PMID: 17274610
ZINC14977010 agonist Compound 17g EC50 = 7.3 nM PMID: 17274610 PPAR_alpha
ZINC14977013 agonist Compound 17h EC50 = 43 nM PMID: 17274610
ZINC14977016 agonist Compound 17i EC50 = 56 nM PMID: 17274610
ZINC14977019 agonist Compound 17j EC50 = 67 nM PMID: 17274610
ZINC14977022 agonist Compound 29f EC50 = 11 nM PMID: 17274610 PPAR_alpha
ZINC14977025 agonist Compound 17k EC50 = 117 nM PMID: 17274610
ZINC14977028 agonist Compound 17l EC50 = 4.6 nM PMID: 17274610 PPAR_alpha
ZINC14977031 agonist Compound 17m EC50 = 2.4 nM PMID: 17274610
ZINC14977034 agonist Compound 17n EC50 = 1.6 nM PMID: 17274610 PPAR_alpha
ZINC14977037 agonist Compound 17o EC50 = 25 nM PMID: 17274610 PPAR_alpha
ZINC14977040 agonist Compound 17p EC50 = 1.9 nM PMID: 17274610
ZINC14977044 agonist Compound 17q EC50 = 7.5 nM PMID: 17274610
ZINC14977051 agonist Compound 17r EC50 = 2.7 nM PMID: 17274610 PPAR_alpha
ZINC14977054 agonist Compound 17s EC50 = 14 nM PMID: 17274610 PPAR_alpha
ZINC14977058 agonist Compound 17t EC50 = 2.2 nM PMID: 17274610
ZINC14977061 agonist Compound 17u EC50 = 11 nM PMID: 17274610
ZINC14977064 agonist Compound 17v EC50 = 367 nM PMID: 17274610 PPAR_alpha
ZINC14977067 agonist Compound 17w EC50 = 2230 nM PMID: 17274610 PPAR_alpha
ZINC14977072 agonist Compound 17x EC50 = 3.4 nM PMID: 17274610 PPAR_alpha
ZINC14977075 agonist Compound 29a EC50 = 5.9 nM PMID: 17274610
ZINC14977078 agonist Compound 29b EC50 = 3.8 nM PMID: 17274610 PPAR_alpha
ZINC14977081 agonist Compound 29c EC50 = 1.5 nM PMID: 17274610 PPAR_alpha
ZINC14977084 agonist Compound 29d EC50 = 2.3 nM PMID: 17274610 PPAR_alpha
ZINC14977087 agonist Compound 29e EC50 = 43 nM PMID: 17274610
ZINC14977091 agonist Compound 29g EC50 = 5.6 nM PMID: 17274610
ZINC14977098 agonist Compound 29h EC50 = 2.2 nM PMID: 17274610 PPAR_alpha
ZINC14977102 agonist Compound 29i EC50 = 0.95 nM PMID: 17274610 PPAR_alpha
ZINC14977105 agonist Compound 34a EC50 = 1.6 nM PMID: 17274610 PPAR_alpha
ZINC14977108 agonist Compound 34b EC50 = 0.58 nM PMID: 17274610 PPAR_alpha
ZINC14977111 agonist Compound 34c EC50 = 2.7 nM PMID: 17274610 PPAR_alpha
ZINC14977114 agonist Compound 34d EC50 = 4.4 nM PMID: 17274610
ZINC14977118 agonist Compound 34e EC50 = 11 nM PMID: 17274610 PPAR_alpha
ZINC14977121 agonist Compound 34f EC50 = 2.5 nM PMID: 17274610 PPAR_alpha
ZINC14977124 agonist Compound 34g EC50 = 11 nM PMID: 17274610 PPAR_alpha
ZINC14977127 agonist Compound 34h EC50 = 3.3 nM PMID: 17274610 PPAR_alpha
ZINC14977130 agonist Compound 34i EC50 = 2.9 nM PMID: 17274610 PPAR_alpha
ZINC14977135 agonist Compound 34j EC50 = 2.9 nM PMID: 17274610 PPAR_alpha
ZINC14977140 agonist Compound 34k EC50 = 4 nM PMID: 17274610 PPAR_alpha
ZINC14977143 agonist Compound 34l EC50 = 1.3 nM PMID: 17274610 PPAR_alpha
ZINC14977146 agonist Compound 34m EC50 = 3.5 nM PMID: 17274610 PPAR_alpha
ZINC14977150 agonist Compound 34n EC50 = 4.1 nM PMID: 17274610 PPAR_alpha
ZINC14977153 agonist Compound 34o EC50 = 2.2 nM PMID: 17274610 PPAR_alpha
ZINC14977156 agonist Compound 34p EC50 = 1.9 nM PMID: 17274610 PPAR_alpha
ZINC14977159 agonist Compound 34q EC50 = 3.3 nM PMID: 17274610 PPAR_alpha
ZINC14977162 agonist Compound 34r EC50 = 4.0 nM PMID: 17274610 PPAR_alpha
ZINC14977165 agonist Compound 34s EC50 = 1.3 nM PMID: 17274610 PPAR_alpha
ZINC14977169 agonist Compound 34u EC50 = 6.9 nM PMID: 17274610 PPAR_alpha
ZINC14977174 agonist Compound 34w EC50 = 3.4 nM PMID: 17274610 PPAR_alpha
ZINC14977178 agonist Compound 34x EC50 = 4.4 nM PMID: 17274610 PPAR_alpha
ZINC14977181 agonist Compound 34y EC50 = 2.1 nM PMID: 17274610 PPAR_alpha
ZINC14977184 agonist Compound 34aa EC50 = 46 nM PMID: 17274610 PPAR_alpha
ZINC14977187 agonist Compound 34ab EC50 = 28 nM PMID: 17274610
ZINC14977190 agonist Compound 34ac EC50 = 12 nM PMID: 17274610 PPAR_alpha
ZINC14977193 agonist Compound 34ae EC50 = 1.3 nM PMID: 17274610 PPAR_alpha
ZINC14977197 agonist Compound 34af EC50 = 3.0 nM PMID: 17274610 PPAR_alpha
ZINC14977200 agonist Compound 34ag EC50 = 1.2 nM PMID: 17274610 PPAR_alpha
ZINC14977203 agonist Compound 34ah EC50 = 2 nM PMID: 17274610 PPAR_alpha
ZINC14977206 agonist Compound 34ai EC50 = 3.4 nM PMID: 17274610 PPAR_alpha
ZINC14977209 agonist Compound 34aj EC50 = 2.3 nM PMID: 17274610 PPAR_alpha
ZINC14977213 agonist Compound 34al EC50 = 3.2 nM PMID: 17274610 PPAR_alpha
ZINC14977216 agonist Compound 34am EC50 = 6 nM PMID: 17274610 PPAR_alpha
ZINC14977219 agonist Compound 34an EC50 = 5.4 nM PMID: 17274610 PPAR_alpha
ZINC15112963 agonist Compound 10 EC50 = 22.6 +/- 1.8 µM PMID: 22381047 PPAR_gamma
ZINC16052148 agonist Compound 10 EC50 = 4.300 µM PMID: 17034149
PPAR_alpha
ZINC16052349 agonist Compound 25a EC50 = 2.83 +/- 1.18 µM PMID: 17243659 PPAR_alpha
ZINC26743888 agonist Compound 19 EC50 = 93 nM PMID: 11677135
PPAR_alpha
ZINC26744992 agonist Compound 20 EC50 = 430 nM PMID: 11677135
PPAR_alpha
ZINC26747370 agonist Compound 21 EC50 = 1000 nM PMID: 11677135
PPAR_alpha
ZINC26747391 agonist Compound 18 EC50 = 160 nM PMID: 11677135
PPAR_alpha
ZINC26749852 agonist Compound 22 EC50 = 1000 nM PMID: 11677135
PPAR_alpha
ZINC27101121 agonist Compound 12 EC50 = 4.68 µM PMID: 15177462 PPAR_gamma
ZINC27101582 agonist Compound 14 EC50 = 1.27 µM PMID: 15177462
PPAR_alpha
ZINC27102276 agonist Compound 18 EC50 = 3.16 µM PMID: 15177462
PPAR_alpha
ZINC27103304 agonist Compound 10 EC50 = 3.31 µM PMID: 15177462
PPAR_alpha
ZINC28123579 agonist Compound 8a EC50 = 2.17 +/- 1.60 µM PMID: 14584939
PPAR_alpha
ZINC28123586 agonist Compound 3 EC50 = 15 µM PMID: 15713415 PPAR_alpha
ZINC28125812 agonist Compound 7 EC50 = 2.08 +/- 1.38 µM PMID: 14584939
PPAR_alpha
ZINC28127637 agonist Compound 1 EC50 = 18 µM PMID: 17379517 
PPAR_alpha
ZINC28130594 agonist Compound 9 EC50 = 19 µM PMID: 15713415 PPAR_alpha
ZINC28131151 agonist Compound 6 EC50 = 1.8 µM PMID: 15713415 PPAR_alpha
ZINC28131157 agonist Compound 7 EC50 = 4.1 µM PMID: 15713415 PPAR_alpha
ZINC28232511 agonist Compound 6f EC50 = 2.0 µM PMID: 11354382 PPAR_alpha
ZINC28235468 agonist Compound 6a EC50 = 1.1 µM PMID: 11354382 PPAR_alpha
ZINC28235832 agonist Compound 6c EC50 = 5.0 µM PMID: 11354382 PPAR_alpha
ZINC28236053 agonist Compound 6h EC50 = 4.0 µM PMID: 11354382 PPAR_alpha
ZINC28569243 agonist Compound 16a EC50 = 12 nM PMID: 16275077
PPAR_alpha
ZINC28569401 agonist Compound 16b EC50 = 23 nM PMID: 16275077
PPAR_alpha
ZINC28569402 agonist Compound 19 EC50 = 700 nM PMID: 16275077 PPAR_alpha
ZINC28604428 agonist Compound 23 EC50 = 4.05 +/- 1.1 µM PMID: 17243659 PPAR_alpha
ZINC28635465 agonist Compound 1 EC50 = 47.6 +/- 4.6 µM PMID: 22381047 PPAR_gamma
ZINC28652276 agonist Compound 5h EC50 = 1.7 +/- 0.1 nM PMID: 17532641
ZINC28652283 agonist Compound (R)-5i EC50 = 3000 +/- 300 nM PMID: 17532641 PPAR_alpha
ZINC28652287 agonist Compound (S)-5i EC50 =1.9 +/- 0.2 nM PMID: 17532641 PPAR_alpha
ZINC28704625 agonist Compound 3S EC50 = 25.0 nM PMID: 17524639
ZINC28704627 agonist Compound 3R EC50 = 1.9 nM PMID: 17524639
ZINC28704665 agonist Compound 7S EC50 = 70.0 nM PMID: 17524639
ZINC28704667 agonist Compound 7R EC50 = 2.1 nM PMID: 17524639
ZINC28704699 agonist Compound 15R EC50 = 0.03 nM PMID: 17524639
ZINC28710190 agonist Compound 21 EC50 = 10 nM PMID: 18155554 PPAR_alpha
ZINC28710191 agonist Compound 22 EC50 = 6 nM PMID: 18155554
PPAR_alpha
ZINC28710192 agonist Compound 23 EC50 = 3 nM PMID: 18155554 PPAR_alpha
ZINC28710193 agonist Compound 24 EC50 = 18 nM PMID: 18155554 PPAR_alpha
ZINC28710194 agonist Compound 36 EC50 = 93 +/- 7 nM PMID: 17608467
ZINC28710197 agonist Compound 76 EC50 = 3 nM PMID: 18155554 PPAR_alpha
ZINC28710198 agonist Compound 77 EC50 = 12 nM PMID: 18155554 PPAR_alpha
ZINC28821850 agonist Compound 56 EC50 = 26 nM PMID: 18155554 PPAR_alpha
ZINC28821851 agonist Compound 57 EC50 = 58 nM PMID: 18155554 PPAR_alpha
ZINC28822316 agonist Compound 14 IC50 = 1.7 nM EC50 = 13 nM PMID: 17498950
ZINC28822317 agonist Compound 15 IC50 = 19 nM EC50 = 252 nM PMID: 17498950
ZINC28822318 agonist Compound 16 IC50 = 20 nM EC50 = 374 nM PMID: 17498950
ZINC28822319 agonist Compound 17 IC50 = 136 nM EC50 = 295 nM PMID: 17498950
ZINC28822322 agonist Compound 13a IC50 = 10 nM EC50 = 251 nM PMID: 17498950
ZINC28822330 agonist Compound 28e IC50 = 1.7 nM EC50 = 70 nM PMID: 17498950
ZINC28822331 agonist Compound 28b IC50 = 10.4 nM EC50 = 230 nM PMID: 17498950
ZINC28822334 agonist Compound 28a IC50 = 286 nM EC50 = 2610 nM PMID: 17498950
ZINC28822682 agonist Compound 10b IC50 = 7.7 nM EC50 = 226 nM PMID: 17512197
ZINC28822697 agonist Compound 10c IC50 = 11 nM EC50 = 305 nM PMID: 17512197
ZINC28822699 agonist Compound 10d IC50 = 14 nM EC50 = 243 nM PMID: 17512197
ZINC28822700 agonist Compound 10e IC50 = 81 nM EC50 = 323 nM PMID: 17512197
ZINC28822702 agonist Compound 10f IC50 = 25 nM EC50 = 1610 nM PMID: 17512197
ZINC28822705 agonist Compound 10h IC50 = 58 nM EC50 = 227 nM PMID: 17512197
ZINC28822706 agonist Compound 10i IC50 = 23 nM EC50 = 638 nM PMID: 17512197
ZINC28822707 agonist Compound 10j IC50 = 37 nM EC50 = 656 nM PMID: 17512197
ZINC28822708 agonist Compound 10k IC50 = 375 nM EC50 = 6360 nM PMID: 17512197
ZINC28822709 agonist Compound 10l IC50 = 37 nM EC50 = 561 nM PMID: 17512197
ZINC28822710 agonist Compound 10m IC50 = 97 nM EC50 = 2630 nM PMID: 17512197
ZINC28822711 agonist Compound 10n IC50 = 244 nM EC50 = 2230 nM PMID: 17512197
ZINC28822712 agonist Compound 10o IC50 = 43 nM EC50 = 172 nM PMID: 17512197
ZINC28822713 agonist Compound 10p IC50 = 15 nM EC50 = 166 nM PMID: 17512197
ZINC28822714 agonist Compound 10q IC50 = 3.6 nM EC50 = 1070 nM PMID: 17512197
ZINC28822715 agonist Compound 10r IC50 = 662 nM EC50 = 3120 nM PMID: 17512197
ZINC28822716 agonist Compound 10s IC50 = 24.1 nM EC50 = 1490 nM PMID: 17512197
ZINC28822717 agonist Compound 10t IC50 = 81 nM EC50 = 3440 nM PMID: 17512197
ZINC28825459 agonist Compound 5 IC50 = 6 nM EC50 = 95 nM PMID: 18029178
PPAR_alpha
ZINC28825460 agonist Compound 6 IC50 = 3 nM EC50 = 38 nM PMID: 18029178
PPAR_alpha
ZINC28825461 agonist Compound 7 IC50 = 4 nM EC50 = 81 nM PMID: 18029178
PPAR_alpha
ZINC28825462 agonist Compound 8 IC50 = 3 nM EC50 = 59 nM PMID: 18029178
PPAR_alpha
ZINC28825463 agonist Compound 9 IC50 = 4 nM EC50 = 22 nM PMID: 18029178
PPAR_alpha
ZINC28825464 agonist Compound 10 IC50 = 3 nM EC50 = 36 nM PMID: 18029178
PPAR_alpha
ZINC28825465 agonist Compound 11 IC50 = 40 nM EC50 = 2870 nM PMID: 18029178 PPAR_gamma
ZINC28825466 agonist Compound 12 IC50 = 32 nM EC50 = 409 nM PMID: 18029178
PPAR_alpha
ZINC28825467 agonist Compound 13 IC50 = 4 nM EC50 = 30 nM PMID: 18029178
PPAR_alpha
ZINC28825468 agonist Compound 14 IC50 = 4 nM EC50 = 286 nM PMID: 18029178
PPAR_alpha
ZINC28825469 agonist Compound 15 IC50 = 6 nM EC50 = 254 nM PMID: 18029178
PPAR_alpha
ZINC28825470 agonist Compound 16 IC50 = 54 nM EC50 = 50 nM PMID: 18029178
PPAR_alpha
ZINC28825471 agonist Compound 17 IC50 = 12 nM EC50 = 376 nM PMID: 18029178
PPAR_alpha
ZINC28825472 agonist Compound 18 IC50 = 64 nM EC50 = 1878 nM PMID: 18029178 PPAR_gamma
ZINC28825473 agonist Compound 19 IC50 = 3 nM EC50 = 96 nM PMID: 18029178
PPAR_alpha
ZINC28825474 agonist Compound 20 IC50 = 5 nM EC50 = 4 nM PMID: 18029178
PPAR_alpha
ZINC28825475 agonist Compound 21 IC50 = 6 nM EC50 = 86 nM PMID: 18029178
PPAR_alpha
ZINC28825476 agonist Compound 22 IC50 = 3 nM EC50 = 48 nM PMID: 18029178
PPAR_alpha
ZINC28825477 agonist Compound 23 IC50 = 3 nM EC50 = 119 nM PMID: 18029178
PPAR_alpha
ZINC28825478 agonist Compound 24 IC50 = 5 nM EC50 = 33 nM PMID: 18029178 PPAR_gamma
ZINC28890851 agonist Compound 7 IC50 = 5 nM EC50 = 6 nM PMID: 17129725 PPAR_gamma
ZINC28890866 agonist Compound 8 IC50 = 8 nM EC50 = 42 nM PMID: 17129725 PPAR_gamma
ZINC28890871 agonist Compound 9 IC50 = 9 nM EC50 = 41 nM PMID: 17129725
PPAR_alpha
ZINC28890877 agonist Compound 10 IC50 = 14 nM EC50 = 399 nM PMID: 17129725
PPAR_alpha
ZINC28890881 agonist Compound 11 IC50 = 3 nM EC50 = 9 nM PMID: 17129725
PPAR_alpha
ZINC28890886 agonist Compound 12 IC50 = 5 nM EC50 = 15 nM PMID: 17129725 PPAR_gamma
ZINC28890891 agonist Compound 13 IC50 = 5 nM EC50 = 5 nM PMID: 17129725 PPAR_gamma
ZINC28890901 agonist Compound 14 IC50 = 3 nM EC50 = 22 nM PMID: 17129725
PPAR_alpha
ZINC28890922 agonist Compound 15 IC50 = 12 nM EC50 = 25 nM PMID: 17129725 PPAR_gamma
ZINC28890927 agonist Compound 16 IC50 = 13 nM EC50 = 274 nM PMID: 17129725
PPAR_alpha
ZINC28890931 agonist Compound 17 IC50 = 5 nM EC50 = 50 nM PMID: 17129725 PPAR_gamma
ZINC28890938 agonist Compound 18 IC50 = 2 nM EC50 = 24 nM PMID: 17129725 PPAR_gamma
ZINC28890943 agonist Compound 19 IC50 = 4 nM EC50 = 6 nM PMID: 17129725
PPAR_alpha
ZINC28890948 agonist Compound 20 IC50 = 3 nM EC50 = 7 nM PMID: 17129725
PPAR_alpha
ZINC28890954 agonist Compound 21 IC50 = 3 nM EC50 = 6 nM PMID: 17129725
PPAR_alpha
ZINC28891480 agonist Compound 11 EC50 = 9 nM PMID: 17157013
ZINC28891487 agonist Compound 12 EC50 = 10 nM PMID: 17157013
ZINC28891492 agonist Compound 14 EC50 = 28 nM PMID: 17157013
ZINC28891497 agonist Compound 15 EC50 = 58 nM PMID: 17157013
ZINC28891503 agonist Compound 16 EC50 = 12 nM PMID: 17157013
ZINC28891508 agonist Compound 17 EC50 = 83 nM PMID: 17157013
ZINC28891516 agonist Compound 18 EC50 = 7 nM PMID: 17157013
ZINC28891521 agonist Compound 19 EC50 = 7 nM PMID: 17157013
ZINC28891546 agonist Compound 20 EC50 = 41 nM PMID: 17157013
ZINC28891551 agonist Compound 21 EC50 = 7 nM PMID: 17157013
ZINC28891564 agonist Compound 22 EC50 = 23 nM PMID: 17157013
ZINC28891589 agonist Compound 23 EC50 = 25 nM PMID: 17157013
ZINC28891599 agonist Compound 24 EC50 = 16 nM PMID: 17157013
ZINC28891605 agonist Compound 25 EC50 = 2 nM PMID: 17157013
ZINC28891622 agonist Compound 26 EC50 = 11 nM PMID: 17157013
ZINC28900607 agonist Compound 20 EC50 = 0.8 µM PMID: 17553678
PPAR_alpha
ZINC28900610 agonist Compound 21 EC50 = 1.4 µM PMID: 17553678
PPAR_alpha
ZINC28900634 agonist Compound 24 R EC50 = 0.002 µM PMID: 17553678
PPAR_alpha
ZINC28900640 agonist Compound 24 S EC50 = 0.13 µM PMID: 17553678
PPAR_alpha
ZINC28900750 agonist Compound 35 R EC50 = 1.19 µM PMID: 17553678
PPAR_alpha
ZINC28900755 agonist Compound 35 S EC50 = 1.57 µM PMID: 17553678
PPAR_alpha
ZINC28900759 agonist Compound 36 R EC50 = 1.58 µM PMID: 17553678
PPAR_alpha
ZINC28900764 agonist Compound 36 S EC50 = 1.80 µM PMID: 17553678
PPAR_alpha
ZINC28902530 agonist Compound 6 EC50 = 2.81 µM PMID: 17524643
ZINC28902543 agonist Compound 9 EC50 = 4.88 µM PMID: 17524643 PPAR_gamma
ZINC28902548 agonist Compound 10 EC50 = 0.94 µM PMID: 17524643 PPAR_gamma
ZINC28902553 agonist Compound 11 EC50 = 1.74 µM PMID: 17524643
ZINC28902558 agonist Compound 12 EC50 = 1.36 µM PMID: 17524643
ZINC28902563 agonist Compound 13 EC50 = 2.61 µM PMID: 17524643
ZINC28902567 agonist Compound 14 EC50 = 2.55 µM PMID: 17524643
ZINC28902571 agonist Compound 15 EC50 = 1.17 µM PMID: 17524643
ZINC28902576 agonist Compound 16 EC50 = 2.97 µM PMID: 17524643
ZINC28902581 agonist Compound 17 EC50 = 0.39 µM PMID: 17524643
ZINC28948386 agonist Compound 2 EC50 = 20 µM PMID: 17379517 
PPAR_alpha
ZINC28948388 agonist Compound 3 EC50 = 1.4 µM PMID: 17379517 
PPAR_alpha
ZINC28948390 agonist Compound 4 EC50 = 13 µM PMID: 17379517 
PPAR_alpha
ZINC28948392 agonist Compound 5 EC50 = 7.9 µM PMID: 17379517 
PPAR_alpha
ZINC28948394 agonist Compound 6 EC50 = 4.0 µM PMID: 17379517 
PPAR_alpha
ZINC28948396 agonist Compound 7 EC50 = 6.0 µM PMID: 17379517 
PPAR_alpha
ZINC28948398 agonist Compound 8 EC50 = 4.0 µM PMID: 17379517 
PPAR_alpha
ZINC28948415 agonist Compound 10 EC50 = 3 µM PMID: 17379517  PPAR_gamma
ZINC28948819 agonist Compound 9 EC50 = 15 µM PMID: 17379517 
PPAR_alpha
ZINC28954798 agonist Compound 1 EC50 = 0.05 µM PMID: 17560785
ZINC28954799 agonist Compound 2 EC50 = 0.13 µM PMID: 17560785
ZINC28978854 agonist Compound 14 EC50 = 0.4 µM PMID: 18060776
PPAR_alpha
ZINC29057355 agonist Compound 79 EC50 = 3 nM PMID: 18155554 PPAR_alpha
ZINC29057646 agonist Compound 75 EC50 = 9 nM PMID: 18155554
PPAR_alpha
ZINC29057804 agonist Compound 66 EC50 = 229 nM PMID: 18155554
ZINC29057808 agonist Compound 70 EC50 = 2 nM PMID: 18155554
PPAR_alpha
ZINC29057968 agonist Compound 62 EC50 = 237 nM PMID: 18155554
ZINC29058101 agonist Compound 55 EC50 = 25 nM PMID: 18155554
PPAR_alpha
ZINC29058105 agonist Compound 50 EC50 = 93 nM PMID: 18155554
ZINC29058241 agonist Compound 45 EC50 = 102 nM PMID: 18155554 PPAR_alpha
ZINC29058249 agonist Compound 40 EC50 = 8 nM PMID: 18155554 PPAR_alpha
ZINC29058367 agonist Compound 30 EC50 = 5 nM PMID: 18155554
PPAR_alpha
ZINC29058372 agonist Compound 35 EC50 = 3 nM PMID: 18155554 PPAR_alpha
ZINC29058615 agonist Compound 20 EC50 = 2 nM PMID: 18155554 PPAR_alpha
ZINC29058739 agonist Compound 13 EC50 = 150 nM PMID: 18155554
ZINC29058743 agonist Compound 16 EC50 = 20 nM PMID: 18155554
ZINC29058747 agonist Compound 10 EC50 = 5 nM PMID: 18155554 PPAR_alpha
ZINC29058857 agonist Compound 6 EC50 = 2 nM PMID: 18155554
ZINC29059179 agonist Compound 86 EC50 = 20 nM PMID: 18155554 PPAR_alpha
ZINC29059200 agonist Compound 82 EC50 = 534 nM PMID: 18155554 PPAR_alpha
ZINC29059206 agonist Compound 83 EC50 = 148 nM PMID: 18155554 PPAR_alpha
ZINC29059402 agonist Compound 80 EC50 = 13 nM PMID: 18155554 PPAR_alpha
ZINC29059409 agonist Compound 81 EC50 = 114 nM PMID: 18155554 PPAR_alpha
ZINC29127122 agonist Compound 13 EC50 = 870 nM PMID: 18162399
PPAR_alpha
ZINC29127161 agonist Compound 12 EC50 = 120 nM PMID: 18162399
PPAR_alpha
ZINC29132176 agonist Compound 20 EC50 (%inhibition) = 20.2 PMID: 18083521
PPAR_alpha
ZINC29132182 agonist Compound 18 EC50 (%inhibition) = 8.4 PMID: 18083521
PPAR_alpha
ZINC29132184 agonist Compound 19 EC50 (%inhibition) = 29.6 PMID: 18083521
PPAR_alpha
ZINC29132261 agonist Compound 16 EC50 (%inhibition) = 17.3 PMID: 18083521
PPAR_alpha
ZINC29132263 agonist Compound 17 EC50 (%inhibition) = 9.6 PMID: 18083521
PPAR_alpha
ZINC29132264 agonist Compound 14 EC50 (%inhibition) = 16.3 PMID: 18083521
PPAR_alpha
ZINC29132266 agonist Compound 15 EC50 (%inhibition) = 19.3 PMID: 18083521
PPAR_alpha
ZINC29132642 agonist Compound 6 EC50 (%inhibition) = 31.3 PMID: 18083521
PPAR_alpha
ZINC29132644 agonist Compound 7 EC50 (%inhibition) = 29.1 PMID: 18083521
PPAR_alpha
ZINC29132646 agonist Compound 8 EC50 (%inhibition) = 22.4 PMID: 18083521
PPAR_alpha
ZINC31157255 agonist Compound 2 EC50 = 53.1 +/- 6.2 µM PMID: 22381047 PPAR_gamma
ZINC32207668 agonist Compound 12 EC50 (%inhibition) = 24.6 PMID: 18083521
PPAR_alpha
ZINC33954913 agonist Compound 12/13 EC50 = 51.1 +/- 5.6 µM PMID: 22381047 PPAR_gamma
ZINC34001583 agonist Compound 4 EC50 = 0.1 µM PMID: 21515063
PPAR_alpha
ZINC34044490 agonist Compound 5 EC50 = 11 µM PMID: 15713415 PPAR_alpha
ZINC34210397 agonist Compound 28 IC50 = 0.892 µM EC50 = 2.2 µM PMID: 16737814
PPAR_alpha
ZINC34251438 agonist Compound 5 EC50 = 0.83 +/- 0.10 µM PMID: 17343371
ZINC34393524 agonist Compound 14a EC50 = 300 +/- 15 nM PMID: 21530275 PPAR_alpha
ZINC34598050 agonist Compound (S)-4f EC50 = 3.0 µM PMID: 22133631 PPAR_alpha
ZINC34717672 agonist Compound 27 IC50 = 0.259 µM EC50 = 1.6 µM PMID: 16737814
PPAR_alpha
ZINC34717700 agonist Compound 18 IC50 = 5 +/- 0 nM EC50 = 73 +/- 6 nM PMID: 16970391
PPAR_alpha
ZINC34717701 agonist Compound 6 IC50 = 6 +/- 0 nM EC50 = 47 +/- 12 nM PMID: 16970391
PPAR_alpha
ZINC34717702 agonist Compound 17 IC50 = 5 +/- 0 nM EC50 = 1 +/- 0 nM PMID: 16970391
PPAR_alpha
ZINC34717703 agonist Compound 19 IC50 = 4 +/- 0 nM EC50 = 34 +/- 0 nM PMID: 16970391
PPAR_alpha
ZINC34717704 agonist Compound 20 IC50 = 4 +/- 1 nM EC50 = 6 +/- 0 nM PMID: 16970391
PPAR_alpha
ZINC34717709 agonist Compound 13 IC50 = 8 +/- 0 nM EC50 = 70 +/- 22 nM PMID: 16970391
PPAR_alpha
ZINC34717711 agonist Compound 15 IC50 = 4 +/- 0 nM EC50 = 8 +/- 3 nM PMID: 16970391
PPAR_alpha
ZINC34717712 agonist Compound 16 IC50 = 5 +/- 0 nM EC50 = 2 +/- 1 nM PMID: 16970391
PPAR_alpha
ZINC34867419 agonist Compound 28 EC50 = 15 nM PMID: 16797985
PPAR_alpha
ZINC35065299 agonist Compound 9 EC50 = 6.980 µM PMID: 17034149
PPAR_alpha
ZINC35246678 agonist Compound 14 EC50 = 0.02 +/- 0.07 µM PMID: 17243659
PPAR_alpha
ZINC35246701 agonist Compound 34 EC50 = 6.26 µM PMID: 17243659 PPAR_alpha
ZINC35246717 agonist Compound 25j EC50 = 0.808 µM PMID: 17243659 PPAR_alpha
ZINC36411196 agonist Compound 29 EC50 = 45.6 nM PMID: 19168353
ZINC36757774 agonist Compound 23 IC50 = 5 nM EC50 = 19 nM PMID: 11677135
PPAR_alpha
ZINC36757831 agonist Compound 2 EC50 = 0.97 µM PMID: 16546385
ZINC36757832 agonist Compound 5 EC50 = 0.56 µM PMID: 16546385
ZINC36757833 agonist Compound 4 EC50= 0.05 µM PMID: 16546385 PPAR_alpha
ZINC36757863 agonist Compound 21a EC50 = 0.004 µM PMID: 16750626 PPAR_alpha
ZINC36757864 agonist Compound 24d EC50 = 0.03 µM PMID: 16750626 PPAR_alpha
ZINC36757865 agonist Compound 23 EC50 = 7 nM PMID: 16797985
PPAR_alpha
ZINC36757866 agonist Compound 22 EC50 = 16 nM PMID: 16797985
PPAR_alpha
ZINC36757867 agonist Compound 21 EC50 = 98 nM PMID: 16797985
PPAR_alpha
ZINC36757868 agonist Compound 16 EC50 = 82 nM PMID: 16797985
PPAR_alpha
ZINC36757869 agonist Compound 5 EC50 = 457 nM PMID: 16797985
PPAR_alpha
ZINC36757871 agonist Compound 12 EC50 = 4.630 µM PMID: 17034149
PPAR_alpha
ZINC36757876 agonist Compound 45 EC50 = 8.24 +/- 1.75 µM PMID: 17243659
PPAR_alpha
ZINC37866897 agonist Compound 24 EC50 = 0.03 µM PMID: 16546385
ZINC37866898 agonist Compound 23 EC50 = 0.04 µM PMID: 16546385
ZINC37866899 agonist Compound 22 EC50 = 0.21 µM PMID: 16546385
ZINC37866900 agonist Compound 21 EC50 = 0.04 µM PMID: 16546385
ZINC37866901 agonist Compound 20 EC50 = 0.09 µM PMID: 16546385
ZINC37866902 agonist Compound 19 EC50 = 0.11 µM PMID: 16546385
ZINC37866903 agonist Compound 18 EC50 = 0.06 µM PMID: 16546385
ZINC37866904 agonist Compound 17 EC50 = 0.07 µM PMID: 16546385
ZINC37866905 agonist Compound 16 EC50 = 0.07 µM PMID: 16546385
ZINC37866906 agonist Compound 15 EC50 = 0.06 µM PMID: 16546385
ZINC37866907 agonist Compound 14 EC50 = 0.56 µM PMID: 16546385
ZINC37866908 agonist Compound 13 EC50 = 0.03 µM PMID: 16546385
ZINC37866909 agonist Compound 12 EC50 = 0.11 µM PMID: 16546385
ZINC37866910 agonist Compound 11 EC50 = 0.49 µM PMID: 16546385
ZINC37866912 agonist Compound 10 EC50 = 0.35 µM PMID: 16546385
ZINC37866913 agonist Compound 9 EC50 = 0.16 µM PMID: 16546385
ZINC37866915 agonist Compound 8 EC50 = 0.54 µM PMID: 16546385
ZINC37866916 agonist Compound 7 EC50 = 0.03 µM PMID: 16546385
ZINC37866917 agonist Compound 6 EC50 = 0.07 µM PMID: 16546385 PPAR_alpha
ZINC37866918 agonist Compound 1 EC50 = 0.01 µM PMID: 16546385
ZINC37866919 agonist Compound 3 EC50 = 0.11 µM PMID: 16546385 PPAR_alpha
ZINC37866926 agonist Compound 15 EC50 = 0.13 µM PMID: 16750626 PPAR_alpha
ZINC37866927 agonist Compound 21d EC50 = 0.26 µM PMID: 16750626
ZINC37866928 agonist Compound 21e EC50 = 0.31 µM PMID: 16750626
ZINC37866929 agonist Compound 24a EC50 = 0.11 µM PMID: 16750626
ZINC37866930 agonist Compound 24b EC50 = 0.09 µM PMID: 16750626 PPAR_alpha
ZINC37866931 agonist Compound 24c EC50 = 2.59 µM PMID: 16750626
ZINC37866932 agonist Compound 24e EC50 = 0.01 µM PMID: 16750626
ZINC37866933 agonist Compound 24f EC50 = 0.08 µM PMID: 16750626
ZINC37866934 agonist Compound 25 EC50 = 3.67 µM PMID: 16750626
ZINC37866935 agonist Compound 26 EC50 = 0.19 µM PMID: 16750626
ZINC37866936 agonist Compound 29a EC50 = 0.03 µM PMID: 16750626
ZINC37866938 agonist Compound 6 EC50 = 1046 nM PMID: 16797985
ZINC37866939 agonist Compound 17j EC50 = 0.06 µM PMID: 16931011
ZINC37866940 agonist Compound 17i EC50 = 0.05 µM PMID: 16931011
ZINC37866941 agonist Compound 17h EC50 = 0.09 µM PMID: 16931011
ZINC37866942 agonist Compound 17g EC50 = 1.07 µM PMID: 16931011
ZINC37866944 agonist Compound 17f EC50 = 0.56 µM PMID: 16931011
ZINC37866946 agonist Compound 17e EC50 = 0.97 µM PMID: 16931011
ZINC37866948 agonist Compound 17d EC50 = 0.07 µM PMID: 16931011
ZINC37866949 agonist Compound 17c EC50 = 0.20 µM PMID: 16931011
ZINC37866951 agonist Compound 17a EC50 = 0.72 µM PMID: 16931011
ZINC37866952 agonist Compound 41 EC50 = 0.66 µM PMID: 17243659 PPAR_alpha
ZINC37866953 agonist Compound 25d EC50 = 5.4 +/- 0.9 µM PMID: 17243659 PPAR_alpha
ZINC37866954 agonist Compound 25c EC50 = 4.6 +/- 0.5 µM PMID: 17243659 PPAR_alpha
ZINC37866959 agonist Compound 2 EC50 = 0.52 +/- 0.02 µM PMID: 17343371
ZINC37866960 agonist Compound 6 EC50 = 2.3 +/- 0.1 µM PMID: 17343371
ZINC37866961 agonist Compound 4 EC50 = 1.1 +/- 0.1 µM PMID: 17343371
ZINC37866962 agonist Compound 3 EC50 = 5.9 +/- 0.5 µM PMID: 17343371
ZINC38139028 agonist Compound 10 Ki = 0.004 µM EC50 = 0.054 µM PMID: 19464171
PPAR_alpha
ZINC38158119 agonist Compound 8b EC50 = 10.50 +/- 2.27 µM PMID: 14584939
PPAR_alpha
ZINC38309475 agonist Compound 18 EC50 = 46.7 nM PMID: 19168353
ZINC38310496 agonist Compound 30 EC50 = 1.060 µM PMID: 18947994
PPAR_alpha
ZINC38320570 agonist Compound 8 EC50 = 1.360 µM PMID: 18947994
PPAR_alpha
ZINC38323523 agonist Compound 25 EC50 = 1.550 µM PMID: 18947994
PPAR_alpha
ZINC40379961 agonist Compound 12 EC50 = 2.700 µM PMID: 18947994
PPAR_alpha
ZINC40380487 agonist Compound 10 EC50 = 2.870 µM PMID: 18947994
PPAR_alpha
ZINC40391278 agonist Compound 16 EC50 = 2.05 µM PMID: 18947994
PPAR_alpha
ZINC40391945 agonist Compound 27 EC50 = 35.4 nM PMID: 19168353
ZINC40392616 agonist Compound 14 EC50 = 1.150 µM PMID: 18947994
PPAR_alpha
ZINC40393734 agonist Compound 6 EC50 = 2.165 µM PMID: 18947994
PPAR_alpha
ZINC40401175 agonist Compound 12 EC50 = 54.3 nM PMID: 19168353
ZINC40401517 agonist Compound 7 EC50 = 216 nM PMID: 19168353
ZINC40401630 agonist Compound 3 EC50 = 65.5 nM PMID: 19168353
ZINC40423329 agonist Compound 5 pIC50 = 8.1 PEC50 = 6.7 PMID: 18722772
ZINC40424157 agonist Compound 36 pIC50 = 7.8 PEC50 = 7.8 PMID: 18722772
ZINC40424310 agonist Compound 33 pIC50 = 8.2 PEC50 = 6.8 PMID: 18722772
ZINC40424339 agonist Compound 22 pIC50 = 8.0 PEC50 = 7.4 PMID: 18722772
ZINC40425282 agonist Compound 24 pIC50 = 7.7 PEC50 = 7.3 PMID: 18722772
ZINC40428667 agonist Compound 13 pIC50 = 8.4 PEC50 = 5.9 PMID: 18722772
ZINC40429259 agonist Compound 20 pIC50 = 8.2 PEC50 = 7.7 PMID: 18722772
ZINC40430131 agonist Compound 28 pIC50 = 7.5 PEC50 = 7.0 PMID: 18722772
ZINC40430607 agonist Compound 27 pIC50 = 7.2 PEC50 = 6.7 PMID: 18722772
ZINC40430870 agonist Compound 31 pIC50 = 7.3 PEC50 = 6.2 PMID: 18722772
ZINC40827704 agonist Compound 25 EC50 = 69.6 nM PMID: 19168353
ZINC40834180 agonist Compound 7b Transactivation = 1.2 PMID: 18805005 PPAR_gamma
ZINC40847207 agonist Compound 4 EC50 = 10 µM PMID: 18947994
PPAR_alpha
ZINC40860845 agonist Compound 26 EC50 = 45.5 nM PMID: 19168353
ZINC40861449 agonist Compound 28 EC50 = 147 nM PMID: 19168353
ZINC40865299 agonist Compound 22 EC50 = 249 nM PMID: 19168353
ZINC40891654 agonist Compound 29 EC50 = 0.035 µM PMID: 18947994
PPAR_alpha
ZINC40892035 agonist Compound 8 EC50 = 238 nM PMID: 19168353
ZINC40894891 agonist Compound 2 EC50 = 711 nM PMID: 19168353
ZINC40894894 agonist Compound 4 EC50 = 49.8 nM PMID: 19168353
ZINC40896724 agonist Compound 9 EC50 = 138 nM PMID: 19168353
ZINC40943237 agonist Compound 11 pIC50 = 7.9 PEC50 = 5.9 PMID: 18722772
ZINC40943239 agonist Compound 12 pIC50 = 7.7 PEC50 = 5.7 PMID: 18722772
ZINC40943241 agonist Compound 8 pIC50 = 8.3 PEC50 = 6.8 PMID: 18722772
ZINC40954668 agonist Compound 2 pIC50 = 7.9 PEC50 = 6.7 PMID: 18722772
ZINC40956316 agonist Compound 29 pIC50 = 8.4 PEC50 = 7.1 PMID: 18722772
ZINC40957231 agonist Compound 21 pIC50 = 8.0 PEC50 = 7.9 PMID: 18722772
ZINC40972730 agonist Compound 17 pIC50 = 7.6 PEC50 = 6.1 PMID: 18722772
ZINC40973244 agonist Compound 26 pIC50 = 8.0 PEC50 = 7.3 PMID: 18722772
ZINC40973797 agonist Compound 12 Ki = 0.016 µM EC50 = 1.1 µM PMID: 19464171
ZINC40974062 agonist Compound 32 pIC50 = 7.7 PEC50 = 7.9 PMID: 18722772
ZINC40974150 agonist Compound 35 pIC50 = 7.9 PEC50 = 7.0 PMID: 18722772
ZINC40975332 agonist Compound 30 pIC50 = 7.8 PEC50 = 6.8 PMID: 18722772
ZINC40975334 agonist Compound 37 Ki = 0.12 µM EC50= 1.5 µM PMID: 19464171 PPAR_gamma
ZINC40975457 agonist Compound 34 pIC50 = 7.9 PEC50 = 6.8 PMID: 18722772
ZINC40975519 agonist Compound 25 pIC50 = 6.8 PEC50 = 6.3 PMID: 18722772
ZINC40975644 agonist Compound 18 pIC50 = 7.8 PEC50 = 6.5 PMID: 18722772
ZINC40976022 agonist Compound 23 pIC50 = 8.0 PEC50 = 7.5 PMID: 18722772
ZINC40976208 agonist Compound 36 Ki = 0.15 µM EC50= 0.90 µM PMID: 19464171 PPAR_gamma
ZINC40976330 agonist Compound 15 pIC50 = 8.0 PEC50 = 6.1 PMID: 18722772
ZINC40976332 agonist Compound 16 pIC50 = 7.8 PEC50 = 6.0 PMID: 18722772
ZINC40979112 agonist Compound 7e Transactivation = 2.2 PMID: 18805005 PPAR_gamma
ZINC42804577 agonist Compound 14 Ki = 0.036 µM EC50 = 2.9 µM PMID: 19464171
ZINC42804863 agonist Compound 20 Ki = 0.006 µM EC50= 0.043 µM PMID: 19464171 PPAR_gamma
ZINC42804868 agonist Compound 21 Ki = 0.005 µM EC50= 0.044 µM PMID: 19464171 PPAR_gamma
ZINC42804942 agonist Compound 25 Ki = 0.006 µM EC50= 1.2 µM PMID: 19464171 PPAR_gamma
ZINC42806443 agonist Compound 34 Ki = 0.66 µM EC50= 3.1 µM PMID: 19464171
ZINC42807188 agonist Compound 26 Ki = 0.009 µM EC50= 0.34 µM PMID: 19464171 PPAR_gamma
ZINC42807442 agonist Compound 15 Ki = 0.047 µM EC50 = 4.1 µM PMID: 19464171
ZINC42807859 agonist Compound 33 Ki = 0.011 µM EC50= 1.2 µM PMID: 19464171 PPAR_gamma
ZINC42834793 agonist Compound 28 Ki = 0.016 µM EC50= 0.68 µM PMID: 19464171 PPAR_gamma
ZINC42835651 agonist Compound 22 Ki = 0.022 µM EC50= 1.4 µM PMID: 19464171 PPAR_gamma
ZINC42851344 agonist Compound 28 EC50 = 2000 nM PMID: 19275963 PPAR_gamma
ZINC42851547 agonist Compound 27 Ki = 0.004 µM EC50= 0.47 µM PMID: 19464171 PPAR_gamma
ZINC42875255 agonist Compound (S)-4l EC50 = 25 +/- 2 nM PMID: 18662876
PPAR_alpha
ZINC42888208 agonist Compound 6 pIC50 = 7.6 PEC50 = 6.3 PMID: 18722772
ZINC42889354 agonist Compound 7 pIC50 = 8.3 PEC50 = 6.8 PMID: 18722772
ZINC42890929 agonist Compound 7d Transactivation = 1.2 PMID: 18805005 PPAR_gamma
ZINC42920692 agonist Compound 23 Ki = 0.002 µM EC50= 0.22 µM PMID: 19464171 PPAR_gamma
ZINC42921106 agonist Compound 25 EC50 = 11.2 +/- 0.45 µM PMID: 19556125
PPAR_alpha
ZINC42921866 agonist Compound 13 Ki = 0.035 µM EC50 =2.2 µM PMID: 19464171
ZINC43022184 agonist Compound 21 EC50 =1.4 +/- 0.38 µM PMID: 19556125
PPAR_alpha
ZINC43277624 antagonist gsk0660 pIC50 = 6.8 pIC50 = 6.5 PMID: 20128594 
ZINC43640915 agonist Compound 5 EC50 (%inhibition) = 8.9 PMID: 18083521
PPAR_alpha
ZINC44280935 agonist Compound 20 EC50 = 500 nM PMID: 19275963
PPAR_alpha
ZINC44359368 agonist Compound (R)-4l EC50 = 180 +/- 10 nM PMID: 18662876
PPAR_alpha
ZINC45355352 antagonist Compound 16 pIC50 = 7.3 pIC50 = 7.1 PMID: 20128594
ZINC45357049 antagonist Compound 10 pIC50 = 6.7 pIC50 = 6.6 PMID: 20128594
ZINC45357936 antagonist Compound 12 PIc50 = 6.5 pIC50 = 6.7 PMID: 20128594
ZINC45358296 antagonist Compound 13 pIC50 = 6.8 pIC50 = 6.7 PMID: 20128594
ZINC45393353 antagonist Compound 15 pIC50 = 6.9 pIC50 = 6.6 PMID: 20128594
ZINC45394247 antagonist Compound 14 pIC50 = 6.9 pIC50 = 6.6 PMID: 20128594
ZINC45495691 agonist Compound 11 Transactivation = 1.4 PMID: 18805005 PPAR_gamma
ZINC45496383 agonist Compound 7a Transactivation = 1.1 PMID: 18805005 PPAR_gamma
ZINC45497359 agonist Compound 7g Transactivation = 2.2 PMID: 18805005 PPAR_gamma
ZINC45505696 agonist Compound 13 EC50 = 5.27 µM PMID: 19301897
PPAR_alpha
ZINC45506275 agonist Compound 16 EC50 = 4.45 µM PMID: 19301897
PPAR_alpha
ZINC45506726 agonist Compound 7c Transactivation = 1.9 PMID: 18805005 PPAR_gamma
ZINC48957410 agonist Compound 25n EC50 = 6.32 µM PMID: 19928766
ZINC49020965 agonist Compound 29a EC50 = 0.06 µM PMID: 19928766
ZINC49021299 agonist Compound 29ae EC50 = 0.01 µM PMID: 19928766
ZINC49021302 agonist Compound 29af EC50 = 0.01 µM PMID: 19928766
ZINC49021465 agonist Compound 25d EC50 = 4.06 µM PMID: 19928766 PPAR_alpha
ZINC49021468 agonist Compound 25f EC50 = 0.34 µM PMID: 19928766 PPAR_alpha
ZINC49021474 agonist Compound 29o EC50 = 0.05 µM PMID: 19928766
ZINC49021949 agonist Compound 38b EC50 = 0.059 µM PMID: 19928766
ZINC49031221 agonist Compound 29m EC50 = 0.02 µM PMID: 19928766
ZINC49031224 agonist Compound 25j EC50 = 0.19 µM PMID: 19928766
ZINC49031578 agonist Compound 46 EC50 = 0.008 µM PMID: 19928766
ZINC49032067 agonist Compound 29p EC50 = 0.11 µM PMID: 19928766
ZINC49032271 agonist Compound 3g EC50 = 53 nM PMID: 19853439
ZINC49032457 agonist Compound 3f EC50 = 400 nM PMID: 19853439
ZINC49032711 agonist Compound 47 EC50 = 0.009 µM PMID: 19928766
ZINC49032857 agonist Compound 29i EC50 = 0.51 µM PMID: 19928766
ZINC49032859 agonist Compound 29j EC50 = 0.72 µM PMID: 19928766
ZINC49032952 agonist Compound 38aa EC50 = 0.007 µM PMID: 19928766
ZINC49033165 agonist Compound 20 EC50 = 0.12 µM PMID: 19928766
ZINC49033169 agonist Compound 40a EC50 = 0.93 µM PMID: 19928766
ZINC49033389 agonist Compound 3k EC50 = 14 nM PMID: 19853439
ZINC49033496 agonist Compound 40p EC50 = 1.30 µM PMID: 19928766
ZINC49033502 agonist Compound 38a EC50 = 0.068 µM PMID: 19928766
ZINC49033534 agonist Compound 12 EC50 = 1.41 µM PMID: 19928766
ZINC49033614 agonist Compound 25g EC50 = 1.39 µM PMID: 19928766
ZINC49033947 agonist Compound 3i EC50 = 45 nM PMID: 19853439
ZINC49033981 antagonist Compound 3a IC50 = 68 nM PMID: 19853439
ZINC49033983 agonist Compound 3b EC50 = 29 nM PMID: 19853439 PPAR_alpha
ZINC49034017 agonist Compound 13 EC50 = 6.36 µM PMID: 19928766
ZINC49034019 agonist Compound 17 EC50 = 0.81 µM PMID: 19928766
ZINC49034093 agonist Compound 25u EC50 = 2.62 µM PMID: 19928766
ZINC49034095 agonist Compound 25v EC50 = 0.13 µM PMID: 19928766
ZINC49034149 agonist Compound 40q EC50 = 0.14 µM PMID: 19928766
ZINC49034173 agonist Compound 25t EC50 = 0.51 µM PMID: 19928766
ZINC49034220 agonist Compound 22 EC50 = 0.66 µM PMID: 19928766
ZINC49034344 agonist Compound 21 EC50 = 0.25 µM PMID: 19928766
ZINC49034831 antagonist Compound 3h IC50 = 10 nM PMID: 19853439
ZINC49034831 agonist Compound 19 EC50 = 11 nM PMID: 20843696
ZINC49035153 agonist Compound 9 EC50 = 5.67 µM PMID: 19928766
ZINC49035427 agonist Compound 29ac EC50 = 0.65 µM PMID: 19928766
ZINC49035452 agonist Compound 29ag EC50 = 0.11 µM PMID: 19928766
ZINC49036299 agonist Compound 25h EC50 = 2.40 µM PMID: 19928766
ZINC49036319 agonist Compound 16 EC50 = 0.10 µM PMID: 19928766
ZINC49036963 agonist Compound 29aa EC50 = 0.05 µM PMID: 19928766
ZINC49037259 agonist Compound 29ab EC50 = 0.01 µM PMID: 19928766
ZINC49045411 agonist Compound 25q EC50 = 0.19 µM PMID: 19928766
ZINC49045871 agonist Compound 29g EC50 = 0.88 µM PMID: 19928766
ZINC49055310 agonist Compound 3l EC50 = 4.9 nM PMID: 19853439
ZINC49109574 agonist Compound 24 EC50 = 1.6 nM PMID: 20843696 PPAR_alpha
ZINC49547509 agonist Compound 25e EC50 = 4.71 µM PMID: 19928766
ZINC49590143 agonist Compound 38g EC50 = 0.018 µM PMID: 19928766
ZINC49774630 agonist Compound 38ae EC50 = 0.003 µM PMID: 19928766
ZINC49774733 agonist Compound 10 EC50 = 3.30 µM PMID: 19928766
ZINC49774737 agonist Compound 35aa EC50 = 0.003 µM PMID: 19928766
ZINC49774796 agonist Compound 35e EC50 = 0.032 µM PMID: 19928766
ZINC49774807 agonist Compound 35j EC50 = 0.063 µM PMID: 19928766
ZINC49774853 agonist Compound 45 EC50 = 0.018 µM PMID: 19928766
ZINC49774863 agonist Compound 38c EC50 =0.017 µM PMID: 19928766
ZINC49774870 agonist Compound 35h EC50 = 0.007 µM PMID: 19928766
ZINC49774877 agonist Compound 40m EC50 = 0.34 µM PMID: 19928766
ZINC49774968 agonist Compound 38ad EC50 = 0.014 µM PMID: 19928766
ZINC49775005 agonist Compound 40s EC50 = 0.062 µM PMID: 19928766
ZINC49775008 agonist Compound 25i EC50 = 0.35 µM PMID: 19928766
ZINC49775068 agonist Compound 35c EC50 = 0.056 µM PMID: 19928766
ZINC49775072 agonist Compound 29e EC50 = 0.02 µM PMID: 19928766
ZINC49775199 agonist Compound 40j EC50 = 0.38 µM PMID: 19928766
ZINC49775280 agonist Compound 19 EC50 = 0.03 µM PMID: 19928766
ZINC49775364 agonist Compound 35a EC50 = 0.331 µM PMID: 19928766
ZINC49775368 agonist Compound 29f EC50 = 0.15 µM PMID: 19928766
ZINC49775414 agonist Compound 40k EC50 = 2.93 µM PMID: 19928766
ZINC49775436 agonist Compound 29c EC50 = 0.07 µM PMID: 19928766
ZINC49775452 agonist Compound 35t EC50 = 0.544 µM PMID: 19928766
ZINC49775480 agonist Compound 29h EC50 = 0.13 µM PMID: 19928766
ZINC49775727 agonist Compound 29k EC50 = 0.01 µM PMID: 19928766
ZINC49777045 agonist Compound 40r EC50 = 0.48 µM PMID: 19928766
ZINC49777254 agonist Compound 29ad EC50 = 0.01 µM PMID: 19928766
ZINC49777284 agonist Compound 38ac EC50 = 0.008 µM PMID: 19928766
ZINC49777854 agonist Compound 44 EC50 = 0.009 µM PMID: 19928766
ZINC49778048 agonist Compound 35k EC50 = 0.010 µM PMID: 19928766
ZINC49778049 agonist Compound 35ac EC50 = 0.004 µM PMID: 19928766
ZINC49778062 agonist Compound 38ah EC50 = 0.001 µM PMID: 19928766
ZINC49778097 agonist Compound 38h EC50 = 0.003 µM PMID: 19928766
ZINC49780201 agonist Compound 35q EC50 = 0.052 µM PMID: 19928766
ZINC49781223 agonist Compound 35p EC50 = 0.410 µM PMID: 19928766
ZINC49781224 agonist Compound 35r EC50 = 0.045 µM PMID: 19928766
ZINC49781271 agonist Compound 35w EC50 = 0.006 µM PMID: 19928766 PPAR_gamma
ZINC49785222 agonist Compound 35n EC50 = 0.013 µM PMID: 19928766
ZINC49785234 agonist Compound 38af EC50 = 0.001 µM PMID: 19928766
ZINC49785235 agonist Compound 35m EC50 = 0.017 µM PMID: 19928766
ZINC49785236 agonist Compound 35f EC50 = 0.035 µM PMID: 19928766
ZINC49785269 agonist Compound 40d EC50 = 1.20 µM PMID: 19928766
ZINC49785293 agonist Compound 35s EC50 = 0.775 µM PMID: 19928766
ZINC49785294 agonist Compound 35d EC50 = 0.120 µM PMID: 19928766
ZINC49785329 agonist Compound 38e EC50 = 0.008 µM PMID: 19928766
ZINC49785395 agonist Compound 40g EC50 = 2.26 µM PMID: 19928766
ZINC49785399 agonist Compound 41 EC50 = 0.011 µM PMID: 19928766
ZINC49785492 agonist Compound 25p EC50 = 0.32 µM PMID: 19928766
ZINC49785525 agonist Compound 29n EC50 = 0.08 µM PMID: 19928766
ZINC49785558 agonist Compound 29b EC50 = 0.04 µM PMID: 19928766
ZINC49785878 agonist Compound 35g EC50 = 0.026 µM PMID: 19928766
ZINC49785899 agonist Compound 29ah EC50 = 0.07 µM PMID: 19928766
ZINC49792537 agonist Compound 25k EC50 = 5.90 µM PMID: 19928766
ZINC49792547 agonist Compound 40f EC50 = 0.02 µM PMID: 19928766
ZINC49792614 agonist Compound 38f EC50 = 0.006 µM PMID: 19928766
ZINC49792665 agonist Compound 35u EC50 = 0.023 µM PMID: 19928766
ZINC49792711 agonist Compound 40l EC50 = 0.74 µM PMID: 19928766
ZINC49792836 agonist Compound 18 EC50 = 0.47 µM PMID: 19928766
ZINC49792971 agonist Compound 40i EC50 = 0.14 µM PMID: 19928766
ZINC49792990 agonist Compound 35o EC50 = 0.030 µM PMID: 19928766
ZINC49793004 agonist Compound 38d EC50 = 0.034 µM PMID: 19928766
ZINC49793135 agonist Compound 43 EC50 = 0.011 µM PMID: 19928766
ZINC49793139 agonist Compound 40h EC50 = 0.23 µM PMID: 19928766
ZINC49793140 agonist Compound 38ab EC50 = 0.055 µM PMID: 19928766
ZINC49799640 agonist Compound 25s EC50 = 0.13 µM PMID: 19928766
ZINC49799645 agonist Compound 38ag EC50 = 0.002 µM PMID: 19928766
ZINC49803976 agonist Compound 35v EC50 = 0.002 µM PMID: 19928766 PPAR_gamma
ZINC49803977 agonist Compound 35ab EC50 = 0.018 µM PMID: 19928766
ZINC49804003 agonist Compound 35ad EC50 = 0.001 µM PMID: 19928766 PPAR_gamma
ZINC49850902 agonist Compound 29q EC50 = 0.25 µM PMID: 19928766
ZINC49864992 agonist Compound 35b EC50 = 0.160 µM PMID: 19928766
ZINC49867778 agonist Compound 32 Ki = 0.028 µM EC50= 0.37 µM PMID: 19464171 PPAR_gamma
ZINC49872280 agonist Compound 31 Ki = 0.036 µM EC50= 0.35 µM PMID: 19464171 PPAR_gamma
ZINC49877890 agonist Compound 30 Ki = 0.12 µM EC50= 1.1 µM PMID: 19464171 PPAR_gamma
ZINC49881838 agonist Compound 9 Ki = 0.008 µM EC50 = 1.9 µM PMID: 19464171
ZINC49881851 agonist Compound 11 Ki = 0.011 µM EC50 = 1.7 µM PMID: 19464171
ZINC49888670 agonist Compound 19 Ki = 0.007 µM EC50= 0.052 µM PMID: 19464171
PPAR_alpha
ZINC49888742 agonist Compound 29 Ki = 0.035 µM EC50= 0.42 µM PMID: 19464171 PPAR_gamma
ZINC49889090 agonist Compound 24 Ki = 0.0006 µM EC50= 2.0 µM PMID: 19464171
ZINC53230851 agonist Compound 2e PMID: 20403648
ZINC53295731 agonist Compound 2i PMID: 20403648
ZINC60325686 agonist Compound 25 EC50 = 2000 nM PMID: 19275963
PPAR_alpha
ZINC64245795 agonist Compound 25 EC50 = 5.7 nM PMID: 20843696
ZINC64251890 agonist Compound 26 EC50 = 220 nM PMID: 20843696 PPAR_alpha
ZINC64466848 agonist Compound 27 EC50 = 76 nM PMID: 20843696 PPAR_alpha
ZINC66099417 agonist Compound 12c EC50 = 0.8 +/- 0.05 µM PMID: 21215640
PPAR_alpha
ZINC66100342 agonist Compound 6a fold induction = 1.58 PMID: 21195611
PPAR_alpha
ZINC66100345 agonist Compound 6b fold induction = 2.78 PMID: 21195611
PPAR_alpha
ZINC66100383 agonist Compound 6d fold induction = 1.68 PMID: 21195611
PPAR_alpha
ZINC66100386 agonist Compound 6e fold induction = 1.23 PMID: 21195611 PPAR_alpha
ZINC66100388 agonist Compound 6f fold induction = 1.62 PMID: 21195611
PPAR_alpha
ZINC66100753 agonist Compound (R)-19 EC50 = 0.0005 µM PMID: 21094606 PPAR_alpha
ZINC66100864 agonist Compound 6g fold induction = 1.31 PMID: 21195611
PPAR_alpha
ZINC66101611 agonist Compound 12a EC50 = 0.01 +/- 0.003 µM PMID: 21215640
PPAR_alpha
ZINC66112736 agonist Compound (S)-18 EC50 = 0.005 µM PMID: 21094606 PPAR_alpha
ZINC66166629 agonist Compound 18a EC50 = 0.3 +/- 0.009 µM PMID: 21215640
PPAR_alpha
ZINC66251285 agonist Compound 20 EC50 = 0.025 µM PMID: 21112784
ZINC66251343 agonist Compound 6h fold induction = 1.46 PMID: 21195611
PPAR_alpha
ZINC66251537 agonist Compound 6i fold induction = 1.25 PMID: 21195611
PPAR_alpha
ZINC66259488 agonist Compound 12f EC50 = 0.7 +/- 0.09 µM PMID: 21215640
PPAR_alpha
ZINC66259489 agonist Compound 17a EC50 = 0.8 +/- 0.07 µM PMID: 21215640
PPAR_alpha
ZINC66262036 agonist Compound 6k fold induction = 1.31 PMID: 21195611
PPAR_alpha
ZINC71296921 agonist Compound 2 pIC50 = 5.9 PEC50 = 6.8 PMID: 21414782
ZINC71297001 agonist Compound 3a (S) pIC50 = 6.2 PEC50 = 6.5 PMID: 21414782
ZINC71297002 agonist Compound 3b (R) pIC50 = 7.6 PEC50 = 7.9 PMID: 21414782
ZINC71317744 agonist Compound 12 pIC50 = 7.9 PEC50 = 8.7 PMID: 21414782
ZINC71331069 agonist Compound 5 EC50 = 0.011 µM PMID: 21515063
PPAR_alpha
ZINC71331954 agonist Compound 14b EC50 = 580 +/- 20 nM PMID: 21530275 PPAR_alpha
ZINC71332043 agonist Compound 12 EC50 = 2.0 µM PMID: 21515063
PPAR_alpha
ZINC71334180 agonist Compound 16 EC50 = 0.7 µM PMID: 21515063
PPAR_alpha
ZINC71340511 agonist Compound 13 EC50 = 0.9 µM PMID: 21515063
PPAR_alpha
ZINC71340668 agonist Compound 10 EC50 = 1.3 µM PMID: 21515063
PPAR_alpha
ZINC71340789 agonist Compound 14c EC50 = 800 +/- 30 nM PMID: 21530275 PPAR_alpha
ZINC71340970 agonist Compound 18 EC50 = 0.021 µM PMID: 21515063
PPAR_alpha
ZINC71341094 agonist Compound 15 EC50 = 1.2 µM PMID: 21515063
PPAR_alpha
ZINC73313429 agonist Compound 4 PMID: 22185225