Compound ID Pharmacological Profile Compound name Binding data Activity data Bibliographic ref Cross-Reactivity
CHEMBL10778 antagonist Compound 10 CAT activity = 5% Bioorg. Med. Chem. Lett.1997,7,11,1483
ZINC03814360 agonist DHT Kd = 0.2 – 0.5 nM T.A. = 0.001 nM PMID: 10077001
ZINC03814420 agonist R1881 Kd = 0.6 nM T.A. = 0.001 nM PMID: 10077001 PR
ZINC00007581 agonist Compound 24 Ki = 16 +/- 2 nM EC50 = 3 +/- 0 nM (Eff=114+/-18%) PMID: 10230629
ZINC00023574 agonist Compound 22 Ki = 11 +/- 3 nM EC50 = 9 +/- 1 nM (Eff=89+/-9%) PMID: 10230629
ZINC13581066 agonist Compound 14 Ki = 9 +/- 1 nM EC50 = 32 +/- 8 nM (Eff=47+/-9%) PMID: 10230629
ZINC03814396 antagonist Compound 16 Ki = 22 +/- 6 nM IC50 = 33 +/- 15 nM (Eff=66+/-4%) PMID: 10230629
ZINC03814404 agonist Compound 13 Ki = 23 nM EC50 = 66 +/- 35 nM (Eff=30+/-8%) PMID: 10230629
ZINC95619129 antagonist 2-hydroxyflutamide Ki = 27 +/- 8 nM IC50 = 15 +/- 2 nM PMID: 10230629 PR
ZINC13581061 antagonist Compound 9 Ki = 8 +/- 2 nM IC50 = 11 +/- 2 nM (55+/-5%) PMID: 10230629
ZINC13581079 agonist Compound 23 Ki = 15 +/- 4 nM EC50 = 10 +/- 2 nM (Eff=39+/-7%) PMID: 10230629
ZINC13581081 agonist Compound 25 Ki = 29 +/- 4 nM EC50 = 20 +/- 5 nM (Eff=64+/-7%) PMID: 10230629
ZINC13581085 agonist Compound 27 Ki = 32 +/- 10 nM EC50 = 16 +/- 5 nM (Eff=69+/-9%) PMID: 10230629
CHEMBL27297 antagonist Compound 4b Ki = 9 +/- 1 nM IC50 = 20 +/- 1 nM (Eff=45 +/- 11%) PMID: 10340624
ZINC28763003 antagonist Compound 6h Ki = 58 nM IC50 =73 +/- 6 nM (Eff=73+/-2%) PMID: 10340624
ZINC28763203 agonist Compound 16 Ki = 8 nM EC50 = 9 +/- 3 nM (Eff=56+/-3%) PMID: 10340624
ZINC28763532 agonist Compound 6j Ki = 8 +/- 2 nM EC50 = 22 +/- 3 nM (Eff=62+/-11%) PMID: 10340624
ZINC28763626 agonist Compound 6l Ki = 27 nM EC50 = 7 +/-3 nM PMID: 10340624
ZINC28763706 agonist Compound 17 Ki = 2 nM EC50 = 3 +/- 1 nM (Eff=107+/-6%) PMID: 10340624
ZINC28763747 agonist Compound 6c Ki = 29 +/- 9 nM EC50 = 19 +/- 4 nM(Eff=63+/-7%) PMID: 10340624
ZINC28764963 agonist Compound 21 Ki = 15 nM EC50 = 2 +/- 0 nM (Eff=86+/-7%) PMID: 10340624
ZINC03814415 agonist norethindrone PMID: 10350363
ZINC27331582 antagonist Compound 8b Ki = 5 nM IC50 = 212 nM (Eff=95%) PMID: 10743937
ZINC27332000 antagonist Compound 7b Ki = 159 nM IC50 =72 nM (Eff=83%) PMID: 10743937
ZINC27408682 antagonist Compound 5c Ki = 84 +/- 22 nM IC50 = 30 +/- 12 nM (Eff=75+/-3%) PMID: 10743937
ZINC27414065 antagonist Compound 6c Ki = 11 nM IC50 = 22 +/- 10 nM (Eff=66/-1%) PMID: 10743937
ZINC27414229 antagonist Compound 22f Ki = 86 +/- 30 nM IC50 = 45 +/- 8 nM (Eff=94+/-3%) PMID: 10743937
ZINC27415171 antagonist Compound 12a Ki = 20 nM IC50 = 63 +/- 23 nM (Eff=98+/-2%) PMID: 10743937
ZINC27415551 antagonist Compound 9 Ki = 22 nM IC50 = 9 +/- 2 nM (Eff=83+/-3%) PMID: 10743937
ZINC02007483 agonist DTIB Ki = 0.71 +/- 0.22 nM PMID: 10966753
ZINC03814409 agonist testosterone Ki = 1.4 +/- 0.4 nM pEC50 = 8.7 +/- 0.2 PMID: 10966753 PMID: 19856921
ZINC03814364 agonist estradiol PMID: 11861974
ZINC04097304 agonist 9-alpha-fluorocortisol PMID: 11906285
ZINC538564 antagonist bicalutamide PMID: 12015321
ZINC03814362 agonist Compound 33 Ki = 0.3 +/- 0.1 nM PMID: 12488554
ZINC13554387 agonist Compound (R)-19 Ki = 2.9 +/- 0.2 nM PMID: 12488554
ZINC03814372 agonist Compound (S)-19 Ki = 123 +/- 27 nM PMID: 12488554
ZINC03814375 agonist Compound 30 Ki = 5.0 +/- 0.6 nM PMID: 12488554
CHEMBL134277 antagonist Compound 18b Ki = 669 +/- 206 nM IC50 = 215 +/- 45 nM (Eff=52+/-2%) PMID: 12954062 MR
CHEMBL336353 antagonist Compound 15 Ki = 819 +/- 423 IC50 = 1500 nM (Eff=60%) PMID: 12954062
CHEMBL413309 antagonist Compound 9a Ki = 1456 +/- 289 nM IC50 = 900 nM (Eff=60%) PMID: 12954062
ZINC03814359 agonist PMID: 14565775
ZINC03814361 agonist PMID: 14565775
ZINC03814418 agonist 5-β-dihydrotestosterone RBA = 137.9008 PMID: 14565775
ZINC03814426 agonist testosterone propionate RBA = 0.1615 PMID: 14565775
ZINC03814428 agonist DHT benzoate RBA = 1.1801 PMID: 14565775
CHEMBL187605 antagonist Compound 13 Ki = 0.040 µM IC50 = 0.774 µM PMID: 15546739
CHEMBL188129 antagonist Compound 15 Ki = 0.062 µM IC50 = 3.32 µM PMID: 15546739
CHEMBL188261 antagonist Compound 19 Ki = 1.40 µM IC50 = 0.78 µM PMID: 15546739
CHEMBL188545 antagonist Compound 16 Ki = 1.03 µM IC50 = 1.33 µM PMID: 15546739
ZINC38468066 antagonist Compound 17 Ki = 0.248 µM IC50 = 2.54 µM PMID: 15546739
CHEMBL189600 antagonist Compound 29 Ki = 0.124 µM IC50 = 0.300 µM PMID: 15546739
CHEMBL362566 antagonist Compound 26 Ki = 0.018 µM IC50 = 0.200 µM PMID: 15546739
ZINC28463952 antagonist Compound 22 Ki = 0.237 µM IC50 = 0.252 µM PMID: 15546739
ZINC34313811 antagonist Compound 32 Ki = 0.073 µM IC50 = 0.060 µM PMID: 15546739
CHEMBL365921 antagonist Compound 28 Ki = 0.041 µM IC50 = 0.588 µM PMID: 15546739
CHEMBL447184 antagonist Compound 31 Ki = 0.693 µM IC50 = 17.9 µM PMID: 15546739
CHEMBL178886 antagonist Compound 3 Ki = 158 nM IC50 = 307 nM PMID: 15603938
CHEMBL184981 antagonist Compound 13 Ki = 83 nM IC50 = 150 nM PMID: 15603938
CHEMBL182412 antagonist Compound 6 Ki = 100 nM IC50 = 196 nM PMID: 15603938
CHEMBL183882 antagonist Compound 8 Ki = 2810 nM IC50 = 658 nM PMID: 15603938
CHEMBL180681 antagonist Compound 11 Ki = 171 nM IC50 = 68 nM PMID: 15603938
CHEMBL188297 antagonist Compound 4 Ki = 5 nM IC50 = 12 nM PMID: 15603938
CHEMBL361445 agonist Compound 5 Ki = 19 nM IC50 = 224 nM PMID: 15603938
CHEMBL369542 agonist Compound 7 Ki = 9 nM IC50 = 49 nM PMID: 15603938
CHEMBL178333 antagonist Compound 16 Ki = 117 nM IC50 = 114 nM PMID: 15603960
CHEMBL178469 antagonist Compound 11 Ki = 632 nM IC50 = 744 nM PMID: 15603960
CHEMBL178957 antagonist Compound 22 Ki = 401 nM IC50 = 1746 nM PMID: 15603960
CHEMBL180859 antagonist Compound 19 Ki = 177 nM IC50 = 517 nM PMID: 15603960
CHEMBL181571 antagonist Compound 21 Ki = 1 nM IC50 > 5 nM PMID: 15603960
CHEMBL181674 antagonist Compound 25 Ki = 11 nM IC50 = 84 nM PMID: 15603960
CHEMBL181722 antagonist Compound 24 Ki = 530 nM IC50 = 1038 nM PMID: 15603960
CHEMBL182186 antagonist Compound 4 Ki = 192 nM IC50 = 664 nM PMID: 15603960
CHEMBL182236 antagonist Compound 18 Ki = 125 nM IC50 = 220 nM PMID: 15603960
CHEMBL359911 antagonist Compound 3 Ki = 284 nM IC50 = 1200 nM PMID: 15603960
CHEMBL361222 agonist Compound 17 Ki = 46 nM IC50 = 146 nM PMID: 15603960
CHEMBL366924 antagonist Compound 20 Ki = 400 nM IC50 = 2014 nM PMID: 15603960
CHEMBL367364 antagonist Compound 13 Ki = 1615 nM IC50 = 317 nM PMID: 15603960
CHEMBL368906 antagonist Compound 14 Ki = 55 nM IC50 = 119 nM PMID: 15603960
CHEMBL197548 antagonist Compound 6 Ki = 2900 nM IC50 = 820 nM PMID: 16019211
CHEMBL198037 antagonist Compound 5 Ki = 3380 nM IC50 = 6800 nM PMID: 16019211
CHEMBL199238 antagonist Compound 9 Ki = 1170 nM IC50 = 7.6 nM PMID: 16019211 VDR
CHEMBL370567 antagonist Compound 8 Ki = 1508 nM IC50 = 9 nM PMID: 16019211 VDR
ZINC03814421 agonist 11-keto-testosterone Kd = 4.44 +/- 1.61 nM PMID: 16107211
ZINC03991694 agonist Compound S-1 Ki = 6.1 nM PMID: 16129672
ZINC04655055 antagonist hydroxyflutamide Ki = 25 nM PMID: 16129672 PR
ZINC13581050 agonist Compound R-3 Ki = 0.3 nM PMID: 16129672
CHEMBL372106 agonist Z-gugulsterone Ki = 315 +/- 13 nM EC50 = 660 +/- 240 nM PMID: 16250653
CHEMBL402063 agonist E-gugulsterone Ki = 240 +/- 21 nM PMID: 16250653
CHEMBL197595 antagonist Compound 33a IC50 = 0.11 µM (Inh=64 +/- 4.3%) PMID: 16420057
CHEMBL200973 antagonist Compound 32 Ki = 4.6 nM IC50 = 0.20 µM (Inh=53 +/- 3.2 %) PMID: 16420057
CHEMBL201069 antagonist Compound 27 IC50 = 0.22 µM (Inh = 36 +/- 5.2 %) PMID: 16420057
CHEMBL201242 antagonist Compound 22 IC50 = 0.13 µM (Inh = 58 +/- 3.5 %) PMID: 16420057
CHEMBL201327 antagonist Compound 30 IC50 = 0.47 µM PMID: 16420057
CHEMBL202710 antagonist Compound 29 IC50 = 0.73 µM (Inh = 52 +/- 3.1 %) PMID: 16420057
CHEMBL202990 antagonist YM-175735 IC50 = 0.20 µM PMID: 16420057
CHEMBL203423 antagonist Compound 18 IC50 = 1.0 µM PMID: 16420057
CHEMBL379465 antagonist Compound 37 IC50 = 0.37 µM (Inh =39 +/- 6.9 %) PMID: 16420057
CHEMBL381253 antagonist Compound 26 IC50 = 0.17 µM (Inh = 52 +/- 4.2 %) PMID: 16420057
CHEMBL439685 antagonist Compound 14 IC50 = 0.12 µM (Inh = 42 +/- 2.2 %) PMID: 16420057
ZINC34886714 antagonist Compound 1b RBA = 6.4 RLA = 0.61 PMID: 16784849
ZINC34886716 antagonist Compound 1h RBA= 12.6 RLA = 0.62 PMID: 16784849
CHEMBL210880 antagonist Compound 44 IC50 (LNCaP) = 0.2 µM PMID: 16789753
CHEMBL212610 antagonist Compound 40 IC50 (LNCaP)= 2.6 µM PMID: 16789753
CHEMBL212693 antagonist Compound 4 IC50  (LNCaP)= 0.2 µM PMID: 16789753
ZINC03874498 antagonist nilutamide IC50 = 4.05 µM PMID: 16857237
CHEMBL217168 antagonist Compound 4c Ki = 153 nM IC50 = 34 +/- 11 nM (Eff=72 +/- 4 %) PMID: 17034117
CHEMBL217324 agonist Compound 4h Ki = 6.3 nM EC50 = 1.9 +/- 0.7 nM (Eff=81 +/- 8 %) PMID: 17034117
CHEMBL217402 agonist Compound 4g Ki = 7.4 nM EC50 = 2.2 +/- 0.4 nM (Eff=77 +/- 13%) PMID: 17034117
CHEMBL217769 agonist Compound 4k Ki = 7.1 nM EC50 = 0.4 +/- 0.1 nM (Eff=107 +/- 5%) PMID: 17034117
CHEMBL267260 agonist Compound 4l Ki = 7.1 nM EC50 = 2.8 +/- 1.6 nM (Eff=99 +/- 13%) PMID: 17034117
CHEMBL277378 agonist Compound 4d Ki = 4.4 nM EC50 = 2.1 +/- 0.3 nM (Eff=94 +/- 19%) PMID: 17034117
CHEMBL442240 agonist Compound 4e Ki = 64 nM EC50 = 1.5 +/- 0.2 nM (Eff=72 +/- 5%) PMID: 17034117
ZINC08585918 agonist BCH IC50 = 163 nM PMID: 17149866
CHEMBL218809 antagonist Compound 4b Ki = 24 nM IC50 = 260 nM PMID: 17181141
CHEMBL218914 agonist Compound (+/-)10b Ki = 5.5 nM EC50 = 6.3 nM (Eff=101%) PMID: 17181141
CHEMBL219198 agonist Compound 7b Ki = 1.5 nM EC50 = 320 nM (Eff=65%) PMID: 17181141
CHEMBL220359 agonist Compound (+)10a Ki = 1.5 nM EC50 = 281 nM (Eff=63%) PMID: 17181141
CHEMBL374121 agonist Compound 7a Ki = 1.7 nM EC50 = 270 nM (Eff=63%) PMID: 17181141
CHEMBL374781 agonist Compound (+/-)10a Ki = 3.5 nM EC50 = 4.4 nM (Eff=96%) PMID: 17181141
CHEMBL384533 agonist Compound 4a Ki = 1.0 nM EC50 = 385 nM (Eff=85%) PMID: 17181141
ZINC13540519 agonist cortisol IC50 = 116 +/- 9.8 µM EC50 = 39.3 +/- 9.7 µM PMID: 17223690 GR
CHEMBL243137 antagonist Compound 9m Ki = 36 +/- 14 nM IC50 = 58 +/- 9 nM (Eff=76 +/- 2%) PMID: 17257838
CHEMBL243351 antagonist Compound 10c Ki = 30 nM IC50 = 42 nM (Eff=79%) PMID: 17257838
CHEMBL244827 antagonist Compound 9a Ki = 83 +/- 7 nM IC50 = 30 +/- 7 nM (Eff=79 +/- 5%) PMID: 17257838
CHEMBL244828 antagonist Compound 9b Ki =29 +/- 9 nM IC50 = 35 +/- 10 nM (Eff=77 +/- 2%) PMID: 17257838
CHEMBL389366 antagonist Compound 9d Ki = 79 +/- 27 nM IC50 = 56 +/- 10nM (Eff=87 +/- 1%) PMID: 17257838
CHEMBL396209 antagonist Compound 13g Ki = 56 nM IC50 = 27 nM (Eff=72%) PMID: 17257838
CHEMBL396732 antagonist Compound 11a Ki = 30 nM IC50 = 76 +/- 7 nM (Eff=75 +/- 1%) PMID: 17257838
CHEMBL441152 antagonist Compound 13e Ki = 74 nM IC50 = 42 +/- 8 nM (Eff=82 +/- 2%) PMID: 17257838
ZINC14968401 agonist Compound 6c Ki = 0.5 nM EC50 = 0.4 +/- 0.1 nM (Eff=74 +/- 7%) PMID: 17267219
ZINC14968405 agonist Compound 6d Ki = 2.3 nM EC50 = 0.4 +/- 0 nM (Eff=110 +/- 7 %) PMID: 17267219
ZINC14968411 agonist Compound 6g Ki = 12 nM EC50 = 1.3 +/- 0.4 nM (Eff=88 +/- 4 %) PMID: 17267219
ZINC14968419 agonist Compound 6i Ki = 2.9 nM EC50 = 0.9 +/- 0.3 nM (Eff=107 +/- 17%) PMID: 17267219
ZINC14968422 agonist Compound 6j Ki = 12 nM EC50 = 1.8 +/- 0.5 nM (Eff=81 +/- 10 %) PMID: 17267219
ZINC14968437 agonist Compound 6m Ki = 1.7 nM EC50 = 0.2 +/- 0.1 nM (Eff=84 +/- 7%) PMID: 17267219
ZINC14968441 agonist Compound 6n Ki = 2.6 nM EC50 = 0.5 +/- 0.1 nM (Eff=88 +/- 14%) PMID: 17267219
ZINC14968445 agonist Compound 6o Ki = 6.0 +/- 1.1 nM EC50 = 1.6 +/- 0.8 nM (Eff=67 +/- 7%) PMID: 17267219
ZINC14968492 agonist Compound 7b Ki = 1.4 nM EC50 = 0.8 +/- 0.3 nM (Eff=93 +/- 5%) PMID: 17267219
ZINC14968500 antagonist Compound 7d Ki = 42 nM IC50 = 36 +/- 15  (Eff=83 +/- 1%) PMID: 17267219
ZINC14968508 agonist Compound7f Ki = 0.4 nM EC50 = 0.5 +/- 0.1 nM (Eff=97 +/- 4%) PMID: 17267219
ZINC14968511 agonist Compound 7g Ki = 0.5 nM EC50 = 0.89 +/- 0.58 nM (Eff=115 +/- 13%) PMID: 17267219
ZINC14968515 agonist Compound 7h Ki = 0.5 nM EC50 = 1.0 +/- 0.0 nM (Eff=125 +/- 22 %) PMID: 17267219
ZINC14968531 agonist Compound 8a Ki = 9.2 nM EC50 = 2.3 +/- 0.7 nM (Eff=86 +/- 5%) PMID: 17267219
ZINC14968544 agonist Compound9 Ki = 12 nM EC50 = 3.2 +/- 1.3 nM (Eff=71 +/- 5%) PMID: 17267219
ZINC03938678 agonist Compound 20 Ki = 2.1 nM EC50 = 0.7 nM PMID: 17292608
ZINC14967191 agonist Compound 1 Ki = 3.2 nM EC50 = 2.3 nM PMID: 17292608
ZINC28704363 agonist Compound 7 Ki = 21 nM EC50 = 6.2 nM PMID: 17292608
ZINC28704370 agonist Compound 9 Ki = 24 nM EC50 = 98 nM PMID: 17292608
ZINC28704373 agonist Compound 11 Ki = 1.5 nM EC50 = 2.8 nM PMID: 17292608
ZINC28704375 agonist Compound 12 Ki = 48 nM EC50 = 345 nM PMID: 17292608
ZINC28704376 agonist Compound 13 Ki = 8.5 nM EC50 = 52 nM PMID: 17292608
ZINC28704378 agonist Compound 14 Ki = 4.5 nM EC50 = 1.7 nM PMID: 17292608
ZINC28704381 agonist Compound 16 Ki = 2.9 nM EC50 = 3.6 nM PMID: 17292608
ZINC28704384 agonist Compound 18 Ki = 3.7 nM EC50 = 487 nM PMID: 17292608
ZINC28704386 agonist Compound 19 Ki = 1.3 nM EC50 = 1.7 nM PMID: 17292608
ZINC28704387 agonist Compound 21 Ki = 1.2 nM EC50 = 0.6 nM PMID: 17292608
ZINC28704389 agonist Compound 22 Ki = 8.0 nM EC50 = 2.2 nM PMID: 17292608
ZINC28704391 agonist Compound 23 Ki = 4.3 nM EC50 = 47 nM PMID: 17292608
ZINC28704393 agonist Compound 24 Ki = 3.0 nM EC50 = 1.0 nM PMID: 17292608
ZINC28704396 agonist Compound 26 Ki = 6.1 nM EC50 = 607 nM PMID: 17292608
ZINC28704398 agonist Compound 27 Ki = 0.7 nM EC50 = 1.7 nM PMID: 17292608
ZINC28704399 agonist Compound 28 Ki = 8.1 nM EC50 = 221 nM PMID: 17292608
ZINC28704403 agonist Compound 30 Ki = 14 nM EC50 = 79 nM PMID: 17292608
ZINC28704405 agonist Compound 31 Ki = 3.3 nM EC50 = 36 nM PMID: 17292608
ZINC28655077 antagonist Compound 15 RBA = 36 % AntiPRolif. Activ. = 97 % PMID: 17336533
ZINC28817160 antagonist Compound 44 PMID: 17337185
ZINC03821119 agonist LGD121071 Ki = 11 +/- 2 nM EC50 = 4.1 +/- 0.9 nM (Eff=100 +/- 7 %) PMID: 17439112
ZINC03875484 agonist fluoxymesterone Ki = 5.7 +/- 0.2 nM EC50 = 0.3 +/- 0.1 nM (Eff= 124 +/- 9%) PMID: 17439112
ZINC14967266 agonist Compound 10b Ki = 1.2 +/- 0.4 nM EC50 = 6.4 +/- 1.7 nM (Eff=92 +/- 8%) PMID: 17439112
ZINC14967270 agonist Compound 10c Ki = 9.6 +/- 7.1 nM EC50 = 2.4 +/- 0.3 nM (Eff=83 +/- 8%) PMID: 17439112
ZINC14967281 agonist Compound 10f Ki = 4.0 +/- 1.0 nM EC50 = 3.5 +/- 1.3 nM (Eff= 88 +/- 5%) PMID: 17439112
ZINC14967285 agonist Compound 12a Ki = 1.6 +/- 0.2 nM EC50= 1.4 +/- 0.3 nM (Eff=68 +/- 5%) PMID: 17439112
ZINC14967289 antagonist Compound 12b Ki = 206 +/- 17 nM IC50 = 244 +/- 44 nM (Eff=90 +/- 2%) PMID: 17439112
ZINC14967304 agonist Compound (-)-10h Ki = 25 +/- 4 nM EC50= 7.8 +/- 0.6 nM (Eff=82 +/- 3%) PMID: 17439112
ZINC14967315 agonist Compound 10 j Ki = 34 +/- 7 nM EC50 = 31 +/- 3 nM (Eff=53 +/- 2%) PMID: 17439112
ZINC14967330 agonist Compound 15a Ki = 113 +/- 50 nM EC50 = 133 +/- 9 nM (Eff=80 +/- 3%) PMID: 17439112
ZINC14967349 agonist Compound 16b Ki = 5.6 +/- 1.6 nM EC50 = 3.9 +/- 2.0 nM (Eff=80 +/- 20%) PMID: 17439112
ZINC14967356 agonist Compound 16c Ki = 4.0 +/- 0.9 nM EC50 = 1.9 +/- 0.3 nM (Eff=65 +/- 5%) PMID: 17439112
ZINC14967372 agonist Compound (R)-16e Ki = 7.1 +/- 1.9 nM EC50 = 1.1 +/- 0.2 nM (Eff=82 +/- 5%) PMID: 17439112
ZINC14967383 agonist Compound (R)-16g Ki = 51 +/- 36 nM EC50 = 5.9 +/- 0.4 nM (Eff=46 +/- 23%) PMID: 17439112
ZINC14967386 agonist Compound (R)-16h Ki = 109 +/- 52 nM EC50 = 27 +/- 13 nM (Eff=65 +/- 15%) PMID: 17439112
ZINC14967390 agonist Compound (R)-27 Ki = 27 nM EC50 = 26 +/- 14 nM (Eff=46 +/- 13%) PMID: 17439112
ZINC14967398 agonist Compound 28 Ki = 16 +/- 11 nM EC50 =14 +/- 4 nM (Eff=75 +/- 5%) PMID: 17439112
ZINC33818834 antagonist ganoderol B PMID: 17499997
ZINC13982538 agonist Compound 11a Ki = 0.9 nM EC50 = 1.8 nM PMID: 17552509
ZINC14967206 agonist Compound 8 Ki = 2 nM EC50 = 15 nM PMID: 17552509
ZINC14967209 agonist Compound 9 Ki = 2.2 nM EC50 = 20 nM PMID: 17552509
ZINC14967213 agonist Compound 10a Ki = 1.5 nM EC50 = 5.2 nM PMID: 17552509
ZINC14967217 agonist Compound 12a Ki = 0.9 nM EC50 = 2.5 nM PMID: 17552509
ZINC14967221 agonist Compound 10b Ki = 4.0 nM EC50 = 87 nM PMID: 17552509
ZINC14967225 agonist Compound 11b Ki =1.6 nM EC50 = 7.1 nM PMID: 17552509
ZINC14967229 agonist Compound 12b Ki =1.9 nM EC50 = 48 nM (Eff=65%) PMID: 17552509
ZINC14967233 agonist Compound10c Ki = 2.9 nM EC50 = 13 nM PMID: 17552509
ZINC14967237 agonist Compound11c Ki = 0.7 nM EC50 = 2.6 nM PMID: 17552509
ZINC14967241 agonist Compound 12c Ki = 1.0 nM EC50 = 2.9 nM PMID: 17552509
ZINC14967244 agonist Compound 11d Ki = 2.3 nM EC50 = 7.4 nM PMID: 17552509
ZINC14967248 agonist Compound 12d Ki = 2.2 nM EC50 = 2.1 nM PMID: 17552509
ZINC14967251 agonist Compound 13 Ki = 23 nM EC50 = 108 nM (Eff= 75%) PMID: 17552509
ZINC14967255 agonist Compound 14 Ki = 0.5 nM EC50 = 2.0 nM PMID: 17552509
CHEMBL233773 agonist Compound 3a Ki = 0.45 nM EC50 = 11.9 nM PMID: 17574413
CHEMBL391770 agonist Compound 4b Ki = 20 nM EC50 = 8962 nM PMID: 17574413
ZINC28822679 agonist Compound 3c Ki = 8.2 nM EC50 = 1251 nM PMID: 17574413
ZINC28822680 agonist Compound 3d Ki = 44 nM EC50 = 3517 nM PMID: 17574413
ZINC28822687 agonist Compound 4c Ki = 14 nM EC50 =7729 nM PMID: 17574413
ZINC00538159 antagonist periciazine Ki = 3.0 µM PMID: 17606915
ZINC19203912 antagonist fluphenazine Ki = 0.8 µM PMID: 17606915
ZINC03945835 agonist Compound 18h EC50 = 1 +/- 0.4 nM (Eff=92 +/- 5%) PMID: 17703938 PR
ZINC28953727 antagonist Compound 16b IC50 = 72 nM (Eff=64%) PMID: 17703938
ZINC28953800 agonist Compound 18o EC50 =20 +/- 16 nM (Eff=74 +/- 5%) PMID: 17703938
ZINC28953810 antagonist Compound 18t IC50 = 45 +/- 10 nM (Eff=88 +/- 2%) PMID: 17703938
ZINC16052389 agonist EM5744 RBA = 525% PMID: 17711855
ZINC14968195 antagonist Compound 4a Ki = 1700 nM IC50 = 25 +/- 20 nM (Eff=58 +/- 7%) PMID: 17887661
ZINC14968204 agonist Compound 4b Ki = 72 nM EC50 = 13 nM (Eff=39 +/- 11%) PMID: 17887661
ZINC14968208 agonist Compound 4c Ki = 19 nM EC50 = 2.6 +/- 0.8 nM (Eff=101 +/-14 %) PMID: 17887661
ZINC14968216 agonist Compound 4e Ki = 70 nM EC50 = 21 +/- 3 nM (Eff=71 +/- 9%) PMID: 17887661
ZINC14968220 agonist Compound 4f Ki = 10 nM EC50 = 12 +/- 0.2 nM (Eff=101 +/- 5%) PMID: 17887661
ZINC14968224 agonist Compound 6a Ki = 1.5 +/- 0.2 nM EC50 = 7.1 +/- 0.4 nM (Eff=109 +/- 13%) PMID: 17887661
ZINC03814430 antagonist spironolactone Ki = 39.4 nM IC50 = 523 nM PMID: 18038968 PMID: 20672822
CHEMBL255216 antagonist Compound 28 Ki = 18 nM IC50 = 88 nM PMID: 18291644
CHEMBL255776 antagonist Compound 2 Ki = 21 nM IC50 = 130 nM PMID: 18291644
CHEMBL257668 antagonist Compound 21 Ki = 3.0 nM IC50 = 16 nM PMID: 18291644
CHEMBL271261 antagonist Compound 26 Ki = 27 nM IC50 = 70 nM PMID: 18291644
CHEMBL271262 antagonist Compound 25 Ki = 17 nM IC50 = 120 nM PMID: 18291644
CHEMBL272509 antagonist Compound 20 Ki = 3.0 nM IC50 = 19 nM PMID: 18291644
CHEMBL403039 antagonist Compound 29 Ki = 17 nM IC50 = 40 nM PMID: 18291644
CHEMBL403061 antagonist Compound 24 Ki = 12 nM IC50 = 20 nM PMID: 18291644
CHEMBL403213 antagonist Compound 23 Ki = 4.0 nM IC50 = 38 nM PMID: 18291644
CHEMBL403214 antagonist Compound 22 Ki = 17 nM IC50 = 11 nM PMID: 18291644
CHEMBL403669 antagonist Compound 18 Ki = 17 nM IC50 = 7.0 nM PMID: 18291644
CHEMBL446626 antagonist Compound 27 Ki = 3.0 nM IC50 = 16 nM PMID: 18291644
ZINC02068322 antagonist Compound 1 Ki = 360 nM IC50 = 152 nM PMID: 18291644
ZINC03948653 antagonist Compound 3 Ki = 40 nM IC50 = 774 nM PMID: 18291644
ZINC29126975 antagonist Compound 14 Ki = 1170 nM IC50 = 2860 nM PMID: 18291644
ZINC29127116 antagonist Compound 12 Ki = 692 nM IC50 = 1150 nM PMID: 18291644
ZINC29127118 antagonist Compound 13 Ki = 1110 nM IC50 = 3310 nM PMID: 18291644
ZINC29127159 antagonist Compound 11 Ki = 77.0 nM IC50 = 500 nM PMID: 18291644
ZINC29127210 antagonist Compound 10 Ki = 486 nM IC50 = 2290 nM PMID: 18291644
ZINC29127216 antagonist Compound 9 Ki = 377 nM IC50 = 480 nM PMID: 18291644
ZINC29127280 antagonist Compound 8 Ki = 221 nM IC50 = 350 nM PMID: 18291644
ZINC29127399 antagonist Compound 7 Ki =53.0 nM IC50 = 670 nM PMID: 18291644
ZINC00899824 antagonist Curcumin EC50 = 35.0 µM PMID: 18316193
ZINC04214779 antagonist Vitamin E succinate EC50 = 38.0 µM PMID: 18316193
ZINC03936191 antagonist asoprisnil IC50 = 6.1 nM PMID: 18318463 PR
ZINC12496366 agonist tetrahydrogestrinone EC50 = 4.3 nM PMID: 18395441
CHEMBL256330 agonist Compound (+/-)-33 Ki = 8.3 +/- 1.6 nM EC50 = 5.9 +/- 1.2 nM (Eff=104 +/- 7 %) PMID: 18400499
ZINC29044405 agonist Compound (+/-)-10 EC50 = 3.2 nM (Eff=61%) PMID: 18400499
ZINC29045788 antagonist Compound (+)-(S)-29b IC50 = 44 nM (Eff=86%) PMID: 18400499
ZINC29045982 antagonist Compound (+)-(S)-28b Ki = 180 nM IC50 = 574 +/- 156 nM (Eff=91 +/- 7%) PMID: 18400499
ZINC34799936 agonist Compound (-)-(R)-21a Ki = 18 nM EC50 = 23 +/- 6 nM (Eff=51 +/- 3%) PMID: 18400499
ZINC13919812 agonist Compound 4c IC50 = 26 nM EC50 = 13 nM PMID: 21944856
ZINC34022720 agonist Compound 1 IC50 = 5.1 nM EC50 = 2.3 nM PMID: 21944856
ZINC03814366 agonist 11-β-hydroxytestosterone PMID: 18514531
CHEMBL480182 antagonist ISOP-4 IC50 = 0.4 µM PMID: 18571420
ZINC40411224 antagonist Compound 54 Ki = 0.37 µM IC50 = 4.9 µM PMID: 18571420
ZINC40411803 antagonist Compound 45 Ki = 0.17 +/- 0.06 µM IC50 = 2.1 +/- 0.1 µM PMID: 18571420
ZINC40412128 antagonist Compound 50 Ki = 0.11 +/- 0.01 µM IC50 = 1.7 +/- 0.1 µM PMID: 18571420
ZINC40412441 antagonist Compound 39 Ki = 0.14 +/- 0.05 µM IC50 = 2.0 +/- 0.8 µM PMID: 18571420
ZINC40412585 antagonist Compound 40 Ki = 0.18 +/- 0.04 µM IC50 = 6.1 +/- 3.1 µM PMID: 18571420
ZINC40413281 antagonist Compound 17 Ki = 2.2 +/- 1.8 µM IC50 = 5.8 +/- 0.2 µM PMID: 18571420
ZINC40414110 antagonist Compound 13 Ki = 2.7 +/- 1.6 µM IC50 = 10 µM PMID: 18571420
ZINC40414183 antagonist Compound 47 Ki = 0.22 µM IC50 = 1.95 µM PMID: 18571420
ZINC40933232 antagonist Compound 26 Ki = 1.8 +/- 0.5 µM IC50 = 5.5 +/- 2.6 µM PMID: 18571420
ZINC40933552 antagonist Compound 53 Ki = 0.34 µM IC50 = 3.7 µM PMID: 18571420
ZINC40934004 antagonist Compound 48 Ki = 0.10 +/- 0.01 µM IC50 = 0.99 +/- 0.59 µM PMID: 18571420
ZINC40934571 antagonist Compound 19 Ki = 2.0 +/- 0.5 µM IC50 = 15.5 +/- 3.5 µM PMID: 18571420
ZINC40935185 antagonist Compound 22 Ki = 0.11 +/- 0.02 µM IC50 = 0.44 +/- 0.08 µM PMID: 18571420
ZINC40935219 antagonist Compound 16 Ki = 0.69 +/- 0.05 µM IC50 = 6.6 +/- 4.8 µM PMID: 18571420
ZINC40935758 antagonist Compound 37 Ki = 0.13 +/- 0.06 µM IC50 = 0.61 +/- 0.23 µM PMID: 18571420
ZINC40936060 antagonist Compound 44 Ki = 0.18 +/- 0.015 µM IC50 = 0.95 +/- 0.28 µM PMID: 18571420
ZINC40936768 antagonist Compound 21 Ki = 0.52 +/- 0.42 µM IC50 = 0.88 +/- 0.18 µM PMID: 18571420
ZINC40981295 antagonist Compound 9 Ki = 3.1 +/- 1.0 µM IC50 = 15.0 +/- 0.2 µM PMID: 18571420
ZINC03812944 antagonist flutamide RBA = 13.7 % IC50 = 58 µM PMID: 18707892
ZINC40379364 antagonist Compound 25 IC50 = 0.73 µM PMID: 19138519
ZINC40407981 antagonist Compound 13 IC50 = 18.9 µM PMID: 19138519
ZINC40845169 antagonist Compound 11 IC50 = 10.0 µM PMID: 19138519
ZINC40859808 antagonist Compound 40 IC50 = 1.9 µM PMID: 19138519
ZINC40898749 antagonist Compound 10 IC50 = 25.8 µM PMID: 19138519
ZINC40914516 antagonist Compound 5 IC50 = 7.7 µM PMID: 19138519
ZINC36435471 antagonist ganoderic acid DM IC50 = 10.6 µM PMID: 19289282
CHEMBL483746 antagonist Compound 11 Ki = 10 +/- 2 nM IC50 = 1800 nM PMID: 19351168
ZINC13982536 agonist Compound 6c Ki = 0.3 +/- 0.1 nM EC50 = 0.2 +/- 0.1 nM PMID: 19351168
ZINC34554150 agonist Compound 6f Ki = 0.3 +/- 0.1 nM EC50 = 1.4 +/- 0.2 nM PMID: 19351168
ZINC40410391 agonist Compound 15 Ki = 17 nM EC50 = 1109 nM PMID: 19351168
ZINC40410424 agonist Compound 6d Ki = 0.2 +/- 0.5 nM EC50 = 19 +/- 3 nM PMID: 19351168
ZINC40412674 agonist Compound 6b Ki = 0.3 +/- 0.1 nM EC50 = 14 +/- 0.5 nM PMID: 19351168
ZINC40420358 agonist Compound 6g Ki = 0.7 +/- 0.2 nM EC50 = 3.7 +/- 0.6 nM PMID: 19351168
ZINC40938487 agonist Compound 6a Ki = 0.8 +/- 0.5 nM EC50 = 4.8 +/- 0.6 nM PMID: 19351168
ZINC40943002 agonist Compound 6e Ki = 2.3 +/- 0.3 nM EC50 = 1.1 +/- 0.1 nM PMID: 19351168
ZINC53195704 agonist Compound 12 Ki = 1.9 +/- 0.1 nM EC50 = 44 nM PMID: 19351168
ZINC34270438 agonist Compound 20 IC50 = 62 nM EC50 = 62 nM (Eff=93%) PMID: 19606870
ZINC38459796 agonist Compound 21 IC50 = 59 nM EC50 = 17 nM (Eff=141%) PMID: 19606870
ZINC38476923 agonist Compound 17 IC50 = 35 nM EC50 = 17 nM (Eff=92%) PMID: 19606870
ZINC38477862 agonist Compound 16 IC50 = 116 nM EC50 = 26 nM (Eff=140%) PMID: 19606870
ZINC62179083 agonist Compound 2 IC50 = 7 nM EC50 = 5 nM (Eff=105%) PMID: 19606870
ZINC42923032 antagonist Compound 1 IC50 (LNCaP)= 20.6 µM PMID: 19725582
ZINC42989367 antagonist Compound 10 IC50 (LNCaP) = 2.3 µM PMID: 19725582
ZINC43014319 antagonist Compound 9 IC50 (LNCaP)= 8.7 µM PMID: 19725582
ZINC43016162 antagonist Compound 11 IC50 (LNCaP) = 8.5 µM PMID: 19725582
ZINC43059632 antagonist Compound 6 IC50 (LNCaP) = 1.3 µM PMID: 19725582
ZINC43076001 antagonist Compound 8 IC50 (LNCaP) = 4.5 µM PMID: 19725582
ZINC43120013 antagonist Compound 3 IC50 (LNCaP) = 6.2 µM PMID: 19725582
ZINC03814395 agonist levonorgestrel EC50 = 0.6635 +/- 0.02237 nM PMID: 19836445
ZINC03814419 agonist norethynodrel EC50 = 34.96 +/- 35.18 nM PMID: 19836445 ER_alpha
ZINC03814422 agonist 17-α-methyltestosterone EC50 = 0.05841 +/- 0.08863 nM PMID: 19836445
ZINC03814429 agonist trenbolone PMID: 20138077
ZINC00001411 antagonist eugenol IC50 = 19 +/- 7 µM PMID: 20226658
ZINC00154632 antagonist raspberry ketone IC50 = 252 +/- 26 µM PMID: 20226658
ZINC00526834 antagonist zingerone IC50 = 153 + / - 8 µM PMID: 20226658
ZINC02558108 antagonist P-hydroxyphenylacetone IC50 = 420 +/- 120 µM PMID: 20226658
ZINC35968242 antagonist Commpound 32-d IC50 = 440 nM IC50 = 190 nM PMID: 20381361
ZINC49781439 antagonist Commpound 18a IC50 = 400 nM IC50 = 64 nM PMID: 20381361
ZINC49781440 antagonist Commpound 24 IC50 = 170 nM IC50 = 64 nM PMID: 20381361
ZINC58502022 antagonist Compound 19 Ki = 84 nM IC50 = 129 nM (Inh=95%) PMID: 20584610
ZINC58502133 antagonist Compound 21 Ki = 36 nM IC50 = 69 nM (Inh=99%) PMID: 20584610
ZINC58502138 antagonist Compound 27 Ki = 98 nM IC50 = 876 nM (Inh=88%) PMID: 20584610
ZINC58502258 antagonist Compound 28 Ki = 40 nM IC50 = 16 nM (Inh=99%) PMID: 20584610
ZINC58502291 antagonist Compound 32 Ki = 12 nM IC50 = 54 nM (Inh=100%) PMID: 20584610
ZINC58506139 antagonist Compound 18 Ki = 14 nM IC50 = 14 nM (Inh=99%) PMID: 20584610
ZINC58506159 antagonist Compound 24 Ki = 6.6 nM IC50 = 9.3 nM (Inh=99%) PMID: 20584610
ZINC58506218 antagonist Compound 22 Ki = 23 nM IC50 = 54 nM (Inh=99%) PMID: 20584610
ZINC58506233 antagonist Compound 20 Ki = 39 nM IC50 = 215 nM (Inh=98%) PMID: 20584610
ZINC58506371 antagonist Compound 23 Ki = 5.7 nM IC50 = 65 nM (Inh=99%) PMID: 20584610
ZINC58506557 antagonist Compound 30 Ki = 56 nM IC50 = 205 nM (Inh=99%) PMID: 20584610
ZINC58506653 antagonist Compound 31 Ki = 16 nM IC50 = 85 nM (Inh=99%) PMID: 20584610
ZINC58511425 antagonist Compound 34 Ki = 93 nM IC50 = 170 nM (Inh=98%) PMID: 20584610
ZINC58512299 antagonist Compound 38 Ki = 3.5 nM IC50 = 11 nM (Inh=98%) PMID: 20584610
ZINC58520321 antagonist Compound 29 Ki = 29 nM IC50 = 39 nM (Inh=99%) PMID: 20584610
ZINC58541168 antagonist Compound 36 Ki = 22 nM IC50 = 37 nM (Inh=99%) PMID: 20584610
ZINC58575413 antagonist Compound 39 Ki = 6.1 nM IC50 = 31 nM (Inh=99%) PMID: 20584610
ZINC58576392 antagonist Compound 37 Ki = 9.4 nM IC50 = 7.4 nM (Inh=96%) PMID: 20584610
ZINC58599325 antagonist Compound 13 Ki = 50 nM IC50 = 873 nM PMID: 20584610
ZINC58599368 antagonist Compound 15 Ki = 14 nM IC50 = 32 nM (Inh=99%) PMID: 20584610
ZINC58602712 antagonist Compound 16 Ki = 37 nM IC50 = 182 nM (Inh=97%) PMID: 20584610
ZINC58602845 antagonist Compound 35 Ki = 9.0 nM IC50 = 7.4 nM (Inh=98%) PMID: 20584610
ZINC58603138 antagonist Compound 25 Ki = 11 nM IC50 = 12 nM (Inh=99%) PMID: 20584610
ZINC58603260 antagonist Compound 26 Ki = 176 nM IC50 = 313 nM (Inh=97%) PMID: 20584610
ZINC58603299 antagonist Compound 17 Ki = 3.7 nM IC50 = 24 nM (Inh=99%) PMID: 20584610
ZINC58655555 antagonist Compound 33 Ki = 32 nM IC50 = 54 nM (Inh=100%) PMID: 20584610
ZINC64361274 antagonist Compound 18 IC50 = 3 µM PMID: 20826091
ZINC28528431 antagonist Compound (R,S)-2 Ki = 1100 nM IC50 = 68 nM PMID: 20888766 VDR
ZINC28528430 antagonist Compound (S,S)-2 Ki = 1100 nM IC50 = 13 nM PMID: 20888766 VDR
ZINC28528433 antagonist Compound (R,R)-2 Ki = 1000 nM IC50 = 14 nM PMID: 20888766 VDR
ZINC28528432 antagonist Compound (S,R)-2 Ki = 1000 nM IC550 = 3.0 nM PMID: 20888766 VDR
ZINC64503983 antagonist Compound 16b IC50 = 0.88 µM PMID: 20888766
ZINC64504070 antagonist Compound 16c IC50 = 0.13 µM PMID: 20888766
ZINC64512502 antagonist Compound 15c IC50 = 9.8 µM PMID: 20888766
ZINC64512813 antagonist Compound (S)-3 Ki = 1800 nM IC50 = 32 nM PMID: 20888766
ZINC64512815 antagonist Compound (R)-3 Ki = 1100 nM IC50 = 15 nM PMID: 20888766
ZINC64513793 antagonist Compound 15b IC50 = 1.1 µM PMID: 20888766 VDR
ZINC64528451 antagonist Compound 16a IC50 = 1.7 µM PMID: 20888766
ZINC00016183 agonist Commpound 23 EC5 = 1.0 nM PMID: 21050768
ZINC34808313 antagonist Commpound 7 IC50 = 200 nM PMID: 21050768
ZINC43197765 antagonist Commpound 17b IC50 = 700 nM PMID: 21050768
ZINC35793633 agonist Compound 2 RBA = 5.5 +/- 1.8 % PMID: 21506597
ZINC66167073 antagonist Compound 7 RBA = 1.84 +/- 0.7 % PMID: 21506597
ZINC71294299 antagonist Compound 8 RBA = 0.37 +/- 0.02 % PMID: 21506597
ZINC71295080 antagonist Compound 6 RBA = 0.97 +/- 0.33 % PMID: 21506597
ZINC73197915 antagonist Compound 4 Inhibition = 50% PMID: 22148427
ZINC03814379 agonist nandrolone PMID: 3865479 ER_alpha
ZINC03814394 agonist gestodene RBA = 33 % PMID: 7750284 PR
ZINC03814382 antagonist mifepristone (RU486) Ki = 10.6 +/- 2.9 nM IC50 = 5 +/- 2 nM (Eff=75 +/- 2%) PMID: 8627601
PR
ZINC03833829 antagonist Compound 27a Ki = 737 +/- 195 nM IC50 = 377 +/- 49 nM (Eff=90 +/- 1%) PMID: 8627601
ZINC03833841 antagonist Compound 22a Ki = 6303 +/- 3708 nM IC50 = 250 nM (Eff=21%) PMID: 8627601
ZINC04428529 antagonist Progesterone Ki = 8.5 +/- 3.1 nM IC50 = 37 +/- 2 nM (Eff=46+/- 7%) PMID: 8627601
PR
ZINC03831956 antagonist Compound 25 Ki = 5831 +/- 4168 IC50 = 946 +/- 419 nM (Eff=90 +/- 4%) PMID: 9464360 GR
ZINC13777087 antagonist Compound 13 Ki = 1856 +/- 251 nM IC50 = 745 +/- 285 nM (Eff=78 +/- 5%) PMID: 9464360
ZINC13777101 antagonist Compound 18 Ki = 1526 +/- 360 IC50 = 253 +/- 156 nM (Eff=88 +/- 8%) PMID: 9464360
ZINC13777103 antagonist Compound 19 Ki = 2138 +/- 341 IC50 = 401 +/- 13 nM (Eff=90 +/- 7%) PMID: 9464360
ZINC13777116 antagonist Compound 24 Ki = 795 +/- 95 IC50 = 315 +/- 42 nM (Eff=90 +/- 5%) PMID: 9464360
ZINC13778369 antagonist Compound 19g Ki = 69 +/- 28 nM IC50 = 48 +/- 4 nM (Eff=85 +/- 1%) PMID: 9484511
ZINC03814399 antagonist Compound 21b Ki = 17 +/- 4 nM IC50 = 19 +/- 3 nM (81+/- 3%) PMID: 9484511 PR
ZINC03814423 antagonist cyproterone acetate Ki = 14 +/- 5 nM IC50 = 26 +/- 23 nM (Eff=48 +/- 6%) PMID: 9484511
ZINC13778335 antagonist Compound 9d Ki = 85 +/- 32 nM IC50 = 22 +/- 4 nM (Eff=78 +/- 2%) PMID: 9484511
ZINC13778356 antagonist Compound 19a Ki = 81 +/- 17 nM IC50 = 34 +/- 6 nM (Eff=89 +/- 2%) PMID: 9484511 PR
ZINC13778384 antagonist Compound 29c Ki = 54 +/- 11 nM IC50 = 27 +/- 7 nM (Eff=49 +/- 7%) PMID: 9484511
ZINC13778395 antagonist Compound 34 Ki = 78 +/- 13 nM IC50 = 27 +/- 5 nM (Eff=85 +/- 2%) PMID: 9484511
ZINC13778399 antagonist Compound 36 Ki = 86 +/- 51 nM IC50 =58 +/- 22 nM (Eff=71 +/- 2%) PMID: 9484511 PR
ZINC13778400 antagonist Compound 42 Ki = 268 +/- 10 nM IC50 = 68 +/- 4 nM (Eff=84 +/- 3%) PMID: 9484511 PR
ZINC03814411 agonist androstanediol PMID: 9736693
ZINC05029557 agonist MPA Ki = 2.9 +/- 0.2 nM EC50 = 6.1 +/- 1.0 nM (Eff=159 +/- 10%) PMID: 9784110 GR
CHEMBL162503 antagonist Compound 5 Ki = 61 +/- 18 nM IC50 = 56 +/- 16 nM (Eff=67 +/- 6%) PMID: 9871534
CHEMBL163366 agonist Compound 8 Ki = 9 +/- 3 nM EC50 = 20 +/- 2 nM (Eff=66 +/- 10%) PMID: 9871534
ZINC03814374 agonist Compound 17 Ki = 4 +/- 1 nM EC50 = 10 +/- 2 nM (Eff=61 +/- 5%) PMID: 9871534
ZINC03814376 agonist Compound 16 Ki = 5 +/- 1 nM EC50 = 5 +/- 1 nM (Eff=91 +/- 6%) PMID: 9871534 PR
ZINC05141582 antagonist Compound 15 Ki = 33 +/- 7 nM IC50 = 56 +/- 8 nM (Eff=82 +/- 2%) PMID: 9871534
ZINC27851181 agonist Compound 9 Ki = 6 +/- 1 nM EC50 = 5 + /- 1 nM (Eff=8 +/- 6%) PMID: 9871534 PR
ZINC27854097 antagonist Compound 6 Ki = 167 +/- 31 nM IC50 = 197 +/- 52 nM (Eff=94 +/- 5%) PMID: 9871534
ZINC27854105 antagonist Compound 29 Ki = 59 nM IC50 = 27 +/- 9 nM (Eff=90 +/- 1%) PMID: 9871534
ZINC49802048 agonist Compound 25 Ki = 9 +/- 2 nM EC50 = 33 +/- 6 nM (Eff=36 +/- 5%) PMID: 9871534
ZINC27854723 agonist Compound 24 Ki = 21 +/- 7 nM EC50 = 25 +/- 2 nM (Eff=60 +/- 9%) PMID: 9871534 PR
ZINC27854781 antagonist Compound 28 Ki = 79 nM IC50 =26 +/- 9 nM (Eff=67 +/- 5%) PMID: 9871534
ZINC27856785 antagonist Compound 18 Ki = 10 +/- 1 nM IC50 = 36 +/- 12 nM (Eff=73 +/- 6%) PMID: 9871534 PR
ZINC22446634 antagonist acetophenazine Ki = 0.8 µM PMID:17606915